SCHEMBL6823722

SCHEMBL6823722

CC(C)(C)[Si](C)(C)Oc1cc([N+](=O)[O-])ccc1N.CC(C)(C)[Si](C)(C)Oc1cc([N+](=O)[O-])ccc1N

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.59
ALDH1A1 P00352 7/20 0.51
TDP1 Q9NUW8 5/20 0.51
CYP3A4 P08684 3/20 0.51
TSHR P16473 2/20 0.46
GAA P10253 1/20 0.42
THRB P10828 1/20 0.42
MAPT P10636 3/20 0.40
RECQL P46063 1/20 0.40
DUSP3 P51452 1/20 0.40
PTPN5 P54829 1/20 0.40
PTPN11 Q06124 1/20 0.40
ALOX15 P16050 1/20 0.40
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 2/20 0.38
RAB9A P51151 1/20 0.38
TLR9 Q9NR96 1/20 0.38
CYP1A2 P05177 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6825987 1.00 HTT (0.59) HTTALDH1A1TDP1CYP3A4TSHR
SCHEMBL16098596 0.90 TDP1 (0.60) HTTALDH1A1TDP1CYP3A4TSHR
SCHEMBL9687587 0.88 HTT (0.46) HTTALDH1A1TDP1CYP3A4TSHR
SCHEMBL62955 0.85 ALDH1A1 (0.50) HTTALDH1A1TDP1CYP3A4TSHR
SCHEMBL2076302 0.84 HTT (0.54) HTTALDH1A1TDP1MAPTMEN1
SCHEMBL1157615 0.84 HTT (0.54) HTTALDH1A1TDP1CYP3A4MAPT
SCHEMBL6823725 0.82 HTT (0.45) HTTALDH1A1CYP3A4TSHRGAA
SCHEMBL61078 0.82 ALDH1A1 (0.51) HTTALDH1A1TDP1CYP3A4TSHR
SCHEMBL18359615 0.81 S1PR4 (0.48) HTTALDH1A1TDP1CYP3A4TSHR
SCHEMBL9172369 0.80 HTT (0.40) HTTALDH1A1TDP1CYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194143-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2004-02-04 EP disclosed
EP-1194143-A2 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2002-04-10 EP disclosed
WO-2000076457-A2 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2000-12-21 WO disclosed
EP-0907362-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-12-01 EP disclosed
EP-0907362-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-04-14 EP disclosed
WO-1997049399-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-12-31 WO disclosed