SCHEMBL6823799

SCHEMBL6823799

COc1cc(Nc2ncnc3cc(O)cc(OC(C)C)c23)ccn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.52
KDR P35968 11/20 0.42
SRC P12931 9/20 0.42
RET P07949 4/20 0.41
KIF5B P33176 3/20 0.41
FGFR1 P11362 1/20 0.41
FLT1 P17948 1/20 0.41
CDK2 P24941 1/20 0.41
PIK3R1 P27986 1/20 0.41
EPHB2 P29323 1/20 0.41
TTBK1 Q5TCY1 1/20 0.41
GAK O14976 1/20 0.41
RIPK2 O43353 1/20 0.41
STK10 O94804 1/20 0.41
FLT3 P36888 1/20 0.41
JAK3 P52333 1/20 0.41
AAK1 Q2M2I8 1/20 0.41
Q6ZSR9 Q6ZSR9 1/20 0.41
SLK Q9H2G2 1/20 0.41
IRAK4 Q9NWZ3 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6819594 0.82 EGFR (0.57) EGFRKDRSRC
SCHEMBL6823640 0.81 EGFR (0.54) EGFRKDRSRCRETLCK
SCHEMBL6831400 0.79 SRC (0.64) EGFRKDRSRCRETKIF5B
SCHEMBL6823586 0.79 SRC (0.61) EGFRKDRSRCRETKIF5B
SCHEMBL6826353 0.77 SRC (0.60) EGFRKDRSRC
SCHEMBL6825683 0.75 SRC (0.74) EGFRKDRSRC
SCHEMBL3280052 0.75 SRC (0.67) EGFRKDRSRCRETKIF5B
SCHEMBL6829839 0.73 SRC (0.60) EGFRKDRSRCRETKIF5B
SCHEMBL6819634 0.73 SRC (0.61) EGFRKDRSRC
SCHEMBL27573718 0.69 KDR (0.48) EGFRKDRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004056812-A1 4- (PYRIDIN-4-YLAMINO) -QUINAZOLINE DERIVATIVES AS ANTI-TUMOR AGENTS ASTRAZENECA AB (SE) 2004-07-08 WO disclosed