SCHEMBL6823928

SCHEMBL6823928

O=C(NC1CCN(CCCCOc2cccc3c2C(=O)/C(=C/CC2CC2)O3)CC1)c1cccc(Cl)c1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 8/20 0.55
HTR1A P08908 4/20 0.55
MCHR1 Q99705 2/20 0.44
CRHR1 P34998 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.40
DRD4 P21917 2/20 0.40
KCNH2 Q12809 1/20 0.40
CACNA1I Q9P0X4 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6820569 1.00 HTR7 (0.55) HTR7HTR1AMCHR1CRHR1L3MBTL1
SCHEMBL6823762 0.92 HTR2A (0.45) HTR7HTR1AMCHR1DRD4
SCHEMBL6823893 0.92 HTR7 (0.45) HTR7HTR1ADRD4
SCHEMBL6823555 0.92 HTR7 (0.45) HTR7HTR1ADRD4
SCHEMBL6823394 0.92 HTR7 (0.45) HTR7HTR1ADRD4
SCHEMBL6824327 0.88 HTR7 (0.42) HTR7HTR1ADRD4KCNH2
SCHEMBL6824547 0.88 HTR7 (0.42) HTR7HTR1ADRD4KCNH2
SCHEMBL6820568 0.83 HTR7 (0.55) HTR7HTR1AMCHR1L3MBTL1DRD4
SCHEMBL6824745 0.80 HTR7 (0.45) HTR7HTR1ADRD4KCNH2POLB
SCHEMBL6823860 0.80 UTS2R (0.49) HTR7HTR1ADRD4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004076444-A2 NOVEL HYDROXYCOUMARANONE DERIVATIVES AS ANTITUMOR AND ANTIMETASTATIC F. HOFFMANN-LA ROCHE AG (CH) 2004-09-10 WO claimed
WO-2004076444-A2 NOVEL HYDROXYCOUMARANONE DERIVATIVES AS ANTITUMOR AND ANTIMETASTATIC F. HOFFMANN-LA ROCHE AG (CH) 2004-09-10 WO disclosed