SCHEMBL6824327

SCHEMBL6824327

NS(=O)(=O)c1cc(C(=O)NC2CCN(CCCCOc3cccc4c3C(=O)/C(=C/CC3CC3)O4)CC2)ccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 5/20 0.42
HTR1A P08908 2/20 0.42
CNR2 P34972 1/20 0.39
UTS2R Q9UKP6 4/20 0.38
DRD4 P21917 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
SSTR5 P35346 1/20 0.38
KCNH2 Q12809 1/20 0.38
ACHE P22303 1/20 0.37
DRD2 P14416 1/20 0.37
HTR2A P28223 1/20 0.37
ADRB1 P08588 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6824547 1.00 HTR7 (0.42) HTR7HTR1ACNR2UTS2RDRD4
SCHEMBL6823555 0.92 HTR7 (0.45) HTR7HTR1AUTS2RDRD4
SCHEMBL6823893 0.92 HTR7 (0.45) HTR7HTR1AUTS2RDRD4
SCHEMBL6823394 0.92 HTR7 (0.45) HTR7HTR1AUTS2RDRD4
SCHEMBL6820569 0.88 HTR7 (0.55) HTR7HTR1ADRD4KCNH2
SCHEMBL6823928 0.88 HTR7 (0.55) HTR7HTR1ADRD4KCNH2
SCHEMBL6823762 0.88 HTR2A (0.45) HTR7HTR1ADRD4DRD2HTR2A
SCHEMBL6826272 0.85 HTR7 (0.47) HTR7HTR1ACNR2UTS2RDRD4
SCHEMBL6378452 0.85 HTR7 (0.46) HTR7HTR1ACNR2UTS2RDRD4
SCHEMBL6824321 0.84 HTR7 (0.46) HTR7HTR1ACNR2UTS2RDRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004076444-A2 NOVEL HYDROXYCOUMARANONE DERIVATIVES AS ANTITUMOR AND ANTIMETASTATIC F. HOFFMANN-LA ROCHE AG (CH) 2004-09-10 WO claimed
WO-2004076444-A2 NOVEL HYDROXYCOUMARANONE DERIVATIVES AS ANTITUMOR AND ANTIMETASTATIC F. HOFFMANN-LA ROCHE AG (CH) 2004-09-10 WO disclosed