SCHEMBL6824958

SCHEMBL6824958

Cc1cccc(C(N)(C(N)=O)c2ccccc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 5/20 0.48
MAPT P10636 1/20 0.47
KMT2A Q03164 1/20 0.47
PARP1 P09874 1/20 0.46
CYP2D6 P10635 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
KCNH2 Q12809 1/20 0.44
POLB P06746 1/20 0.42
KCNN4 O15554 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
HTR3A P46098 1/20 0.41
HTR3D Q70Z44 1/20 0.41
HTR3C Q8WXA8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28091404 0.84 KMT2A (0.52) KIF11MAPTKMT2ACYP2D6POLB
SCHEMBL8169066 0.83 MAPT (0.58) MAPTKMT2APARP1CYP2D6CYP2C19
SCHEMBL16162191 0.79 LMNA (0.51) KIF11MAPTKMT2APARP1CYP2D6
SCHEMBL6825078 0.79 KMT2A (0.43) KIF11MAPTKMT2ACYP2D6KCNN4
SCHEMBL4593887 0.78 PARP1 (0.52) KIF11MAPTKMT2APARP1CYP2D6
SCHEMBL13724829 0.77 MKNK1 (0.43) MAPTKMT2APARP1CYP3A4SMN1; SMN2
SCHEMBL5744305 0.77 LMNA (0.55) KIF11MAPTKMT2APARP1CYP2D6
SCHEMBL27621135 0.77 KMT2A (0.62) KIF11MAPTKMT2APARP1CYP2D6
SCHEMBL27438603 0.76 PARP1 (0.46) KIF11MAPTKMT2APARP1CYP3A4
SCHEMBL4232590 0.76 MAPK1 (0.48) KIF11MAPTPARP1CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004022534-A1 ARYLGLYCINE DERIVATIVES FOR USE AS GLYCINE TRANSPORT INHIBITORS NPS ALLELIX CORP. (CA) 2004-03-18 WO disclosed