SCHEMBL4593887

SCHEMBL4593887

Cc1cccc(C(C(N)=O)(C(N)=O)c2cccc(C)c2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.52
HTR3E A5X5Y0 2/20 0.46
HTR3B O95264 2/20 0.46
HTR3A P46098 2/20 0.46
HTR3D Q70Z44 2/20 0.46
HTR3C Q8WXA8 2/20 0.46
KIF11 P52732 5/20 0.45
LMNA P02545 2/20 0.45
MAPT P10636 1/20 0.44
KMT2A Q03164 1/20 0.44
KCNN4 O15554 1/20 0.43
ACHE P22303 2/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KCNH2 Q12809 1/20 0.41
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
PTPN5 P54829 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7841877 0.87 ACHE (0.53) PARP1HTR3EHTR3BHTR3AHTR3D
SCHEMBL27621135 0.82 KMT2A (0.62) PARP1HTR3EHTR3BHTR3AHTR3D
SCHEMBL5744305 0.82 LMNA (0.55) PARP1HTR3EHTR3BHTR3AHTR3D
SCHEMBL30087612 0.81 PARP1 (0.48) PARP1HTR3EHTR3BHTR3AHTR3D
SCHEMBL27438603 0.78 PARP1 (0.46) PARP1HTR3EHTR3BHTR3AHTR3D
SCHEMBL16162191 0.78 LMNA (0.51) PARP1HTR3EHTR3BHTR3AHTR3D
SCHEMBL6824958 0.78 KIF11 (0.48) PARP1HTR3EHTR3BHTR3AHTR3D
SCHEMBL16892960 0.76 KCNN4 (0.72) PARP1KIF11MAPTKMT2AKCNN4
SCHEMBL16892944 0.76 PARP1 (0.52) PARP1HTR3EHTR3BHTR3AHTR3D
SCHEMBL16892940 0.76 CES2 (0.55) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116693529-A Synthesis method of 2-aza [2.2.2] octane compound 河南师范大学 2023-09-05 CN disclosed
EP-1937257-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES Nederlandse Organisatie voor toegepast- natuurwetenschappelijk onderzoek TNO (NL) 2008-07-02 EP disclosed
WO-2007037685-A1 NOVEL ANTIBIOTICS COMPRISING BIS(1-ARYL-5-TETRAZ0LYL)METHANE DERIVATIVES NEDERLANDSE ORGANISATIE VOOR TOEGEPAST-NATUURWETENSCHAPPELIJK ONDERZOEK TNO (NL) 2007-04-05 WO disclosed