SCHEMBL6826837

SCHEMBL6826837

COc1nnc(Cl)cc1C(N)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 3/20 0.43
ALDH1A1 P00352 5/20 0.41
LMNA P02545 1/20 0.41
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NNMT P40261 4/20 0.40
POLB P06746 2/20 0.39
SYK P43405 1/20 0.38
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
KDM4E B2RXH2 3/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
PRNP P04156 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
PPARG P37231 1/20 0.36
HTT P42858 1/20 0.36
MAPK10 P53779 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17141437 0.84 POLB (0.43) ALDH1A1LMNARAB9AL3MBTL1POLB
SCHEMBL1750237 0.84 ALDH1A1 (0.46) CASP1ALDH1A1LMNARAB9AL3MBTL1
SCHEMBL15633425 0.82 KDM4E (0.46) ALDH1A1LMNARAB9AL3MBTL1POLB
SCHEMBL24158869 0.80 NNMT (0.45) CASP1ALDH1A1NNMTPOLBROCK2
SCHEMBL1751822 0.79 HMGCR (0.44) ALDH1A1LMNARAB9AL3MBTL1POLB
SCHEMBL25228251 0.78 ALDH1A1 (0.39) ALDH1A1LMNARAB9AL3MBTL1POLB
SCHEMBL669037 0.75 CASP1 (0.56) CASP1ALDH1A1LMNARAB9AL3MBTL1
SCHEMBL12611466 0.74 NNMT (0.46) CASP1ALDH1A1LMNARAB9ANNMT
SCHEMBL24342278 0.73 IKBKB (0.42) CASP1ALDH1A1LMNANNMTSYK
SCHEMBL16853382 0.73 SYK (0.41) CASP1ALDH1A1LMNARAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004108707-A1 PYRIDAZINIL QUINAZOLINE DERIVATIVES FOR USE IN THE TREATMENT OF TUMOURS ASTRAZENECA AB (SE) 2004-12-16 WO disclosed