SCHEMBL6827151

SCHEMBL6827151

CCOC(=O)CSc1nc(Cl)cc(Cl)n1

nearest known ligand 0.71

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.58
ALOX5 P09917 2/20 0.56
LMNA P02545 1/20 0.56
MAPT P10636 1/20 0.53
ABCB1 P08183 2/20 0.52
TDP1 Q9NUW8 1/20 0.52
ALOX15 P16050 1/20 0.52
ALDH1A1 P00352 2/20 0.52
GAA P10253 2/20 0.52
HPGD P15428 1/20 0.52
HSD17B10 Q99714 1/20 0.52
TSHR P16473 1/20 0.51
KMT2A Q03164 2/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
RXFP1 Q9HBX9 2/20 0.50
MEN1 O00255 1/20 0.50
MAPK1 P28482 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6562061 0.90 L3MBTL1 (0.61) KDM4EALOX5LMNAMAPTABCB1
SCHEMBL11840409 0.86 ALOX5 (0.59) KDM4EALOX5LMNAMAPTABCB1
SCHEMBL13752163 0.84 KDM4E (0.60) KDM4ELMNAMAPTABCB1TDP1
SCHEMBL6565776 0.84 L3MBTL1 (0.70) ALOX5MAPTABCB1TDP1ALDH1A1
SCHEMBL28468685 0.83 GAA (0.63) KDM4ELMNAABCB1TDP1ALOX15
SCHEMBL17085323 0.83 KDM4E (0.54) KDM4ELMNAMAPTABCB1TDP1
SCHEMBL13401380 0.82 KDM4E (0.59) KDM4ELMNAABCB1TDP1ALOX15
SCHEMBL11838953 0.82 LMNA (0.52) KDM4EALOX5LMNAMAPTABCB1
SCHEMBL6565628 0.81 PPARA (0.72) KDM4EALOX5MAPTABCB1ALOX15
SCHEMBL6563326 0.81 ALOX5 (0.61) KDM4EALOX5LMNATDP1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004054988-A1 ARYLTHIOETHERPYRIMIDINE AND ARYLOXYETHERPYRIMIDINE DERIVATIVES AND THEIR THERAPEUTIC USES ACTIVE PASS PHARMACEUTICALS, INC. (CA) 2004-07-01 WO disclosed
EP-0073328-A1 Novel pyrimidine and s. triazine derivatives with antilipidemic activity LPB Istituto Farmaceutico s.p.a. (IT) 1983-03-09 EP disclosed
US-3940394-A ANTILIPEMIC SANTILLI ARTHUR A 1976-02-24 US disclosed