SCHEMBL6827181

SCHEMBL6827181

C[C@]1([C@H](O)c2ccc(-c3ccc4cc(O)ccc4c3)cc2)NC(=O)NC1=O

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 11/20 0.44
ESR2 Q92731 11/20 0.44
ABL1 P00519 2/20 0.39
ABCB1 P08183 2/20 0.39
BCR P11274 2/20 0.39
HSD17B1 P14061 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2B6 P20813 1/20 0.38
CYP2C19 P33261 1/20 0.38
HSD17B2 P37059 1/20 0.38
FTO Q9C0B1 1/20 0.37
PTGER3 P43115 1/20 0.36
CYP17A1 P05093 2/20 0.35
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6827189 1.00 ESR1 (0.44) ESR1ESR2ABL1ABCB1BCR
SCHEMBL6792396 0.89 PTGER3 (0.46) ESR1ESR2HSD17B1HSD17B2PTGER3
SCHEMBL8337588 0.83 FASN (0.38) ABL1PTGER3
SCHEMBL6824386 0.82 CA2 (0.41) PTGER3CYP11B1CYP11B2
SCHEMBL6824389 0.82 CA2 (0.41) PTGER3CYP11B1CYP11B2
SCHEMBL6791153 0.80 MMP2 (0.41) CYP3A4CYP2D6CYP2C9
SCHEMBL6789361 0.80 MMP2 (0.41) CYP3A4CYP2D6CYP2C9
SCHEMBL6791227 0.80 MMP2 (0.41) CYP3A4CYP2D6CYP2C9
SCHEMBL6789612 0.80 PGR (0.36)
SCHEMBL6793983 0.79 MMP2 (0.45) ESR2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004024060-A2 METALLOPROTEINASE INHIBITORS AND INTERMEDIATES FOR PREPARATION THEREOF ASTRAZENECA AB (SE) 2004-03-25 WO claimed
WO-2004024060-A2 METALLOPROTEINASE INHIBITORS AND INTERMEDIATES FOR PREPARATION THEREOF ASTRAZENECA AB (SE) 2004-03-25 WO disclosed
WO-2004024060-A2 METALLOPROTEINASE INHIBITORS AND INTERMEDIATES FOR PREPARATION THEREOF ASTRAZENECA AB (SE) 2004-03-25 WO disclosed