SCHEMBL6827422

SCHEMBL6827422

CC(=O)Oc1ccccc1C(=O)Oc1ccccc1C(=O)OCc1ccc2nc(N)nc(N)c2c1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
HSD17B10 Q99714 1/20 0.48
DHFR P00374 1/20 0.47
MAPT P10636 1/20 0.45
PTGS2 P35354 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6821942 0.99 DHFR (0.48) KDM4ELMNACYP1A2CYP2C9HSD17B10
SCHEMBL6827444 0.90 TDP1 (0.49) KDM4EHSD17B10DHFRMAPT
SCHEMBL6827375 0.84 DHFR (0.47) DHFRMAPT
SCHEMBL6748619 0.83 DHFR (0.52) DHFR
SCHEMBL6827626 0.83 TDP1 (0.56) KDM4EDHFRMAPT
SCHEMBL6747477 0.82 DHFR (0.51) DHFR
SCHEMBL6750825 0.80 DHFR (0.49) DHFR
SCHEMBL6827408 0.80 KDM4E (0.44) KDM4ELMNACYP1A2CYP2C9HSD17B10
SCHEMBL6744730 0.79 DHFR (0.50) DHFR
SCHEMBL6825657 0.78 DHFR (0.41) KDM4ELMNACYP1A2CYP2C9HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004020417-A1 2,4-DIAMINOQUINAZOLINE, 2-AMINO-4-HYDROXYPTERIDINE AND 2,4-DIAMINOPYRIMIDINE ESTER DERIVATIVES AS DIHYDROFOLATE REDUCTASE INHIBITORS MELACURE THERAPEUTICS AB (SE) 2004-03-11 WO claimed
WO-2004020417-A1 2,4-DIAMINOQUINAZOLINE, 2-AMINO-4-HYDROXYPTERIDINE AND 2,4-DIAMINOPYRIMIDINE ESTER DERIVATIVES AS DIHYDROFOLATE REDUCTASE INHIBITORS MELACURE THERAPEUTICS AB (SE) 2004-03-11 WO disclosed