SCHEMBL6828653

SCHEMBL6828653

COC(=O)c1ccc(COc2ccc(Cl)c(Cl)c2)s1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 3/20 0.64
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
LMNA P02545 1/20 0.45
DAO P14920 1/20 0.42
SCN9A Q15858 3/20 0.42
HRH3 Q9Y5N1 1/20 0.42
NOTUM Q6P988 1/20 0.41
SCN5A Q14524 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6826144 0.84 MRGPRX4 (0.78) MRGPRX4TP53
SCHEMBL6826427 0.82 MRGPRX4 (0.56) MRGPRX4ALDH1A1LMNAMEN1KMT2A
SCHEMBL7131595 0.82 MRGPRX4 (0.57) MRGPRX4LMNATP53
SCHEMBL7128455 0.80 MRGPRX4 (0.55) MRGPRX4KDM4ELMNATP53
SCHEMBL6829550 0.80 MRGPRX4 (0.54) MRGPRX4ALDH1A1LMNAMEN1KMT2A
SCHEMBL6829566 0.80 MRGPRX4 (0.54) MRGPRX4ALDH1A1LMNAMEN1KMT2A
SCHEMBL6619558 0.79 MRGPRX4 (0.56) MRGPRX4KDM4EALDH1A1LMNAMEN1
SCHEMBL7129725 0.79 MRGPRX4 (0.54) MRGPRX4HRH3MEN1KMT2A
SCHEMBL22480846 0.78 MRGPRX4 (1.00) MRGPRX4KDM4EKMT2A
SCHEMBL6829631 0.77 RAB9A (0.57) MRGPRX4ALDH1A1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004037808-A1 2 - SUBSTITUTED HETEROCYCLIC COMPOUNDS AND ANTITUMOR COMPOSITION COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2004-05-06 WO disclosed