SCHEMBL6829550

SCHEMBL6829550

COC(=O)c1ccc(COc2ccc(F)cc2)s1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 2/20 0.54
FFAR1 O14842 3/20 0.47
TP53 P04637 1/20 0.45
MAOB P27338 2/20 0.44
MAPT P10636 1/20 0.43
HDAC4 P56524 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
NR4A2 P43354 1/20 0.42
NPSR1 Q6W5P4 2/20 0.42
LMNA P02545 1/20 0.42
PPARG P37231 1/20 0.42
NCOA2 Q15596 1/20 0.42
NCOA1 Q15788 1/20 0.42
NCOA3 Q9Y6Q9 1/20 0.42
NPC1 O15118 1/20 0.42
HSP90AA1 P07900 1/20 0.42
RAB9A P51151 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6826427 0.88 MRGPRX4 (0.56) MRGPRX4FFAR1TP53MAPTHDAC4
SCHEMBL6829566 0.86 MRGPRX4 (0.54) MRGPRX4FFAR1TP53MAOBMAPT
SCHEMBL6619558 0.85 MRGPRX4 (0.56) MRGPRX4TP53MAPTNR4A2NPSR1
SCHEMBL7131595 0.85 MRGPRX4 (0.57) MRGPRX4TP53MAOBMAPTHDAC4
SCHEMBL6829631 0.83 RAB9A (0.57) MRGPRX4FFAR1MAPTHDAC4HDAC6
SCHEMBL6831135 0.81 MRGPRX4 (0.55) MRGPRX4TP53MAPTHDAC4HDAC6
SCHEMBL6828653 0.80 MRGPRX4 (0.64) MRGPRX4TP53LMNAALDH1A1MEN1
SCHEMBL16812822 0.78 MRGPRX4 (0.57) MRGPRX4TP53MAPTHDAC4HDAC6
SCHEMBL7128455 0.78 MRGPRX4 (0.55) MRGPRX4TP53MAOBLMNANPC1
SCHEMBL7129725 0.77 MRGPRX4 (0.54) MRGPRX4FFAR1MAOBMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004037808-A1 2 - SUBSTITUTED HETEROCYCLIC COMPOUNDS AND ANTITUMOR COMPOSITION COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2004-05-06 WO disclosed