SCHEMBL6831129

SCHEMBL6831129

NC(=O)c1cccnc1Sc1ccc(F)c(F)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
SMN1; SMN2 Q16637 3/20 0.47
GAA P10253 1/20 0.47
HTT P42858 2/20 0.43
MAPT P10636 1/20 0.43
CA2 P00918 2/20 0.43
CA4 P22748 2/20 0.43
DDB1 Q16531 1/20 0.43
CRBN Q96SW2 1/20 0.43
KMT2A Q03164 1/20 0.41
LMNA P02545 3/20 0.41
PARP1 P09874 1/20 0.41
ATM Q13315 1/20 0.40
GRM5 P41594 1/20 0.40
KDM4E B2RXH2 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CRHBP P24387 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28040764 0.80 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2GAAMAPTDDB1
SCHEMBL5087696 0.79 SMN1; SMN2 (0.61) ALDH1A1SMN1; SMN2GAADDB1CRBN
SCHEMBL6831130 0.72 SIRT3 (0.43) HTTCA2CA4KMT2AKDM4E
SCHEMBL30680404 0.72 SMN1; SMN2 (0.54) ALDH1A1SMN1; SMN2GAAHTTDDB1
SCHEMBL10827952 0.72 SMN1; SMN2 (0.54) ALDH1A1SMN1; SMN2GAAHTTDDB1
SCHEMBL1327237 0.71 KMT2A (0.56) ALDH1A1HTTKMT2ALMNAPARP1
SCHEMBL5717691 0.70 CRHBP (0.68) ALDH1A1SMN1; SMN2GAAMAPTDDB1
SCHEMBL447126 0.68 NAPRT (0.68) ALDH1A1SMN1; SMN2HTTMAPTLMNA
SCHEMBL31078773 0.68 NAPRT (0.68) ALDH1A1SMN1; SMN2HTTMAPTLMNA
SCHEMBL14040985 0.68 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2GAAMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087669-A1 NOVEL QUINOLINE, TETRAHYDROQUINAZOLINE, AND PYRIMIDINE DERIVATIVES AND METHODS OF TREATMENT RELATED TO THE USE THEREOF TAISHO PHARMACEUTICAL CO. LTD. (JP) 2004-10-14 WO disclosed