SCHEMBL6832655

SCHEMBL6832655

Brc1ccc(CNCCc2ccccc2)cn1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.58
MAPT P10636 1/20 0.58
HDAC1 Q13547 3/20 0.53
BCHE P06276 5/20 0.53
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA4 P22748 1/20 0.48
CA9 Q16790 1/20 0.48
ROCK2 O75116 1/20 0.47
KCNH2 Q12809 1/20 0.47
ROCK1 Q13464 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
SIGMAR1 Q99720 3/20 0.46
TDP1 Q9NUW8 1/20 0.46
OPRM1 P35372 2/20 0.45
OPRD1 P41143 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12854771 0.81 MAOA (0.45) HDAC1ALDH1A1KCNH2TDP1
SCHEMBL6508504 0.80 DRD4 (0.64) GAAHDAC1ROCK1
SCHEMBL11881258 0.78 GAA (0.91) GAAMAPTBCHEKDM4EALDH1A1
SCHEMBL3272134 0.78 GAA (0.91) GAAMAPTBCHEKDM4EALDH1A1
SCHEMBL23642329 0.78 CD274 (0.48) ALDH1A1MEN1KMT2A
SCHEMBL7995688 0.78 CYP11B1 (0.38) HDAC1MEN1KMT2ATDP1
SCHEMBL9511528 0.78 MC4R (0.45) HDAC1SIGMAR1
SCHEMBL6832125 0.78 GAA (0.74) GAAMAPTBCHEKDM4EALDH1A1
SCHEMBL4468862 0.78 GAA (0.74) GAAMAPTBCHEKDM4EALDH1A1
SCHEMBL27228 0.76 GAA (0.95) GAAMAPTBCHEKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096771-A1 BIARYL COMPOUNDS HAVING ACTIVITY AT THE 5HT5A RECEPTOR GLAXO GROUP LIMITED (GB) 2004-11-11 WO disclosed