SCHEMBL6833560

SCHEMBL6833560

CCc1cc(=O)oc2cc(O)c(O)cc12

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 7/20 0.74
AKR1B1 P15121 2/20 0.68
HSD17B3 P37058 2/20 0.65
ALDH1A1 P00352 7/20 0.62
HPGD P15428 6/20 0.62
KDM4E B2RXH2 5/20 0.62
HSD17B10 Q99714 5/20 0.62
CYP3A4 P08684 1/20 0.62
THRB P10828 1/20 0.62
TSHR P16473 1/20 0.58
GAA P10253 4/20 0.57
CASP1 P29466 3/20 0.57
CASP7 P55210 3/20 0.57
GLA P06280 2/20 0.57
POLB P06746 2/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
HTT P42858 2/20 0.54
MAPK1 P28482 1/20 0.54
PPARG P37231 1/20 0.54
MAPK10 P53779 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6836133 0.88 MCL1 (0.68) MCL1AKR1B1HSD17B3ALDH1A1HPGD
SCHEMBL14925273 0.88 MCL1 (0.67) MCL1AKR1B1HSD17B3ALDH1A1HPGD
SCHEMBL13058664 0.86 HSD17B3 (0.58) MCL1AKR1B1HSD17B3ALDH1A1HPGD
SCHEMBL8706801 0.85 MCL1 (1.00) MCL1AKR1B1HSD17B3ALDH1A1HPGD
SCHEMBL6836134 0.85 ALDH1A1 (0.69) MCL1AKR1B1HSD17B3ALDH1A1HPGD
SCHEMBL27527191 0.84 ALDH1A1 (0.63) MCL1AKR1B1HSD17B3ALDH1A1HPGD
SCHEMBL8706946 0.84 MCL1 (0.72) MCL1AKR1B1HSD17B3ALDH1A1HPGD
SCHEMBL13353968 0.84 MCL1 (0.72) MCL1AKR1B1HSD17B3ALDH1A1HPGD
SCHEMBL8702627 0.84 MCL1 (1.00) MCL1AKR1B1HSD17B3ALDH1A1HPGD
SCHEMBL8704051 0.84 MCL1 (0.72) MCL1AKR1B1HSD17B3ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6750249-B1 GRADUALLY RELEASE ESCULETIN OR ITS DERIVATIVE IN A CONTROLLED MANNER OVER A LONG PERIOD OF TIME KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 2004-06-15 US disclosed
EP-1121931-A1 CONTROLLED RELEASE ORAL PREPARATIONS OF ESCULETIN AND ITS DERIVATIVES Kureha Chemical Industry Co., Ltd. (JP) 2001-08-08 EP disclosed
EP-0654479-B1 Esculetin derivatives and method for manufacture thereof, use thereof, and pharmaceutical composition KUREHA CHEMICAL IND CO LTD (JP) 2000-03-15 EP disclosed
US-5736522-A Esculetin derivatives and method for manufacture thereof, use thereof, and pharmaceutical composition KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1998-04-07 US disclosed
EP-0654479-A2 Esculetin derivatives and method for manufacture thereof, use thereof, and pharmaceutical composition KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1995-05-24 EP disclosed