SCHEMBL6836133

SCHEMBL6836133

CCCc1cc(=O)oc2cc(O)c(O)cc12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 7/20 0.68
HSD17B3 P37058 2/20 0.68
AKR1B1 P15121 2/20 0.62
ALDH1A1 P00352 10/20 0.61
TSHR P16473 2/20 0.61
ALDH1A2 O94788 1/20 0.61
ALDH2 P05091 1/20 0.61
MAPT P10636 1/20 0.61
ALDH1B1 P30837 1/20 0.61
ALDH1A3 P47895 1/20 0.61
KDM4E B2RXH2 8/20 0.58
HPGD P15428 6/20 0.58
HSD17B10 Q99714 5/20 0.58
POLB P06746 2/20 0.58
HTT P42858 1/20 0.57
CYP3A4 P08684 1/20 0.57
THRB P10828 1/20 0.57
GAA P10253 4/20 0.56
ERAP1 Q9NZ08 1/20 0.56
SMN1; SMN2 Q16637 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6836134 0.90 ALDH1A1 (0.69) MCL1HSD17B3AKR1B1ALDH1A1TSHR
SCHEMBL27527191 0.89 ALDH1A1 (0.63) MCL1HSD17B3AKR1B1ALDH1A1TSHR
SCHEMBL6833560 0.88 MCL1 (0.74) MCL1HSD17B3AKR1B1ALDH1A1TSHR
SCHEMBL15082519 0.88 HSD17B3 (0.61) MCL1HSD17B3AKR1B1ALDH1A1TSHR
SCHEMBL15082515 0.88 MCL1 (0.61) MCL1HSD17B3ALDH1A1TSHRALDH1A2
SCHEMBL18032945 0.88 ALDH1A1 (0.62) MCL1HSD17B3AKR1B1ALDH1A1TSHR
SCHEMBL15082517 0.85 HSD17B3 (0.58) MCL1HSD17B3AKR1B1ALDH1A1TSHR
SCHEMBL8807721 0.85 HSD17B3 (0.58) MCL1HSD17B3AKR1B1ALDH1A1TSHR
SCHEMBL8702449 0.85 MCL1 (0.75) MCL1HSD17B3AKR1B1ALDH1A1KDM4E
SCHEMBL27508630 0.83 MCL1 (0.68) MCL1HSD17B3AKR1B1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6750249-B1 GRADUALLY RELEASE ESCULETIN OR ITS DERIVATIVE IN A CONTROLLED MANNER OVER A LONG PERIOD OF TIME KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 2004-06-15 US disclosed
EP-1121931-A1 CONTROLLED RELEASE ORAL PREPARATIONS OF ESCULETIN AND ITS DERIVATIVES Kureha Chemical Industry Co., Ltd. (JP) 2001-08-08 EP disclosed
EP-0654479-B1 Esculetin derivatives and method for manufacture thereof, use thereof, and pharmaceutical composition KUREHA CHEMICAL IND CO LTD (JP) 2000-03-15 EP disclosed
US-5736522-A Esculetin derivatives and method for manufacture thereof, use thereof, and pharmaceutical composition KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1998-04-07 US disclosed
EP-0654479-A2 Esculetin derivatives and method for manufacture thereof, use thereof, and pharmaceutical composition KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1995-05-24 EP disclosed