SCHEMBL6836134

SCHEMBL6836134

CCCCc1cc(=O)oc2cc(O)c(O)cc12

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.69
GAA P10253 5/20 0.69
ERAP1 Q9NZ08 1/20 0.69
MCL1 Q07820 6/20 0.64
KDM4E B2RXH2 9/20 0.61
MEN1 O00255 2/20 0.61
KMT2A Q03164 2/20 0.61
MAPK1 P28482 1/20 0.61
MAPT P10636 3/20 0.59
HTT P42858 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
AKR1B1 P15121 2/20 0.59
HSD17B3 P37058 2/20 0.56
HPGD P15428 6/20 0.54
HSD17B10 Q99714 5/20 0.54
CYP3A4 P08684 1/20 0.54
THRB P10828 1/20 0.54
GLA P06280 1/20 0.52
CASP1 P29466 1/20 0.52
CASP7 P55210 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27527191 0.95 ALDH1A1 (0.63) ALDH1A1GAAERAP1MCL1KDM4E
SCHEMBL18032945 0.94 ALDH1A1 (0.62) ALDH1A1GAAERAP1MCL1KDM4E
SCHEMBL6836133 0.90 MCL1 (0.68) ALDH1A1GAAERAP1MCL1KDM4E
SCHEMBL6833560 0.85 MCL1 (0.74) ALDH1A1GAAMCL1KDM4EMEN1
SCHEMBL8702449 0.82 MCL1 (0.75) ALDH1A1GAAERAP1MCL1KDM4E
SCHEMBL30696150 0.82 MCL1 (0.60) ALDH1A1GAAERAP1MCL1KDM4E
SCHEMBL18009960 0.82 MCL1 (0.60) ALDH1A1GAAERAP1MCL1KDM4E
SCHEMBL27508630 0.81 MCL1 (0.68) ALDH1A1GAAERAP1MCL1KDM4E
SCHEMBL15082519 0.79 HSD17B3 (0.61) ALDH1A1GAAERAP1MCL1KDM4E
SCHEMBL15082515 0.79 MCL1 (0.61) ALDH1A1GAAERAP1MCL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6750249-B1 GRADUALLY RELEASE ESCULETIN OR ITS DERIVATIVE IN A CONTROLLED MANNER OVER A LONG PERIOD OF TIME KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 2004-06-15 US disclosed
EP-1121931-A1 CONTROLLED RELEASE ORAL PREPARATIONS OF ESCULETIN AND ITS DERIVATIVES Kureha Chemical Industry Co., Ltd. (JP) 2001-08-08 EP disclosed
EP-0654479-B1 Esculetin derivatives and method for manufacture thereof, use thereof, and pharmaceutical composition KUREHA CHEMICAL IND CO LTD (JP) 2000-03-15 EP disclosed
US-5736522-A Esculetin derivatives and method for manufacture thereof, use thereof, and pharmaceutical composition KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1998-04-07 US disclosed
EP-0654479-A2 Esculetin derivatives and method for manufacture thereof, use thereof, and pharmaceutical composition KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1995-05-24 EP disclosed