SCHEMBL6833701

SCHEMBL6833701

NC(=S)Nc1ncc(Br)cc1CCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
NPC1 O15118 1/20 0.43
KCNH2 Q12809 1/20 0.43
NR3C2 P08235 1/20 0.39
MAPT P10636 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
PKM P14618 1/20 0.39
ALOX12 P18054 2/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
RAB9A P51151 1/20 0.37
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
GCK P35557 1/20 0.36
MGLL Q99685 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TP53 P04637 1/20 0.36
TYR P14679 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2334248 0.78 GCK (0.56) ALDH1A1NPC1KCNH2GCK
SCHEMBL1329926 0.72 NPC1 (0.44) ALDH1A1NPC1KCNH2MAPTMEN1
SCHEMBL1327994 0.72 GCK (0.54) ALDH1A1NPC1KCNH2MAPTALOX12
SCHEMBL2317274 0.72 MAPT (0.55) ALDH1A1NPC1KCNH2MAPTMEN1
SCHEMBL9390463 0.68 MAPT (0.58) ALDH1A1NPC1MAPTALOX12LMNA
SCHEMBL2337875 0.68 MAPKAPK2 (0.40) ALDH1A1KCNH2MEN1KMT2AGCK
SCHEMBL14471918 0.67 NPC1 (0.39) ALDH1A1NPC1KCNH2MAPTMEN1
SCHEMBL6905303 0.66 ALDH1A1 (0.71) ALDH1A1NPC1MAPTMEN1KMT2A
SCHEMBL6901408 0.65 NPC1 (0.51) ALDH1A1NPC1KCNH2MAPTMEN1
SCHEMBL17388766 0.64 CCNE1 (0.51) ALDH1A1NPC1MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10647735-B2 Metal complexes and methods of preparing the same UNIVERSITY OF NEW BRUNSWICK (CA) 2020-05-12 US disclosed
US-20200017535-A1 METAL COMPLEXES AND METHODS OF PREPARING THE SAME UNIVERSITY OF NEW BRUNSWICK (CA) 2020-01-16 US disclosed
US-20040171652-A1 Antiviral and spermicidal contraceptives; 2-thiourea pyridinyl derivative containing compositions PARKER HUGHES INSTITUTE 2004-09-02 US disclosed
US-6774139-B1 CONTRACEPTIVES PARKER HUGHES INSTITUTE 2004-08-10 US disclosed
CN-1371367-A Phenethyl-5-bromopyridylthiourea (PBT) and Dihydroalkoxybenzyloxopyrimidine (DABO) derivatives exhibiting spermicidal activity PARKER HUGHES INST (US) 2002-09-25 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10647735-B2 Metal complexes and methods of preparing the same CACYBP, CLTB, VDAC2 ALDH1A1 4328/4885NPC1 3355/4885KCNH2 167/4885
US-20200017535-A1 METAL COMPLEXES AND METHODS OF PREPARING THE SAME CACYBP, CLTB, VDAC2 ALDH1A1 4328/4885NPC1 3355/4885KCNH2 167/4885
US-20040171652-A1 Antiviral and spermicidal contraceptives; 2-thiourea pyridinyl derivative containing compositions ZP1, NASP, SAMHD1 ALDH1A1 1417/4885NPC1 4052/4885KCNH2 2772/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.