SCHEMBL6836622

SCHEMBL6836622

CS(=O)(=O)Oc1ccc(-c2sc3cc(OS(=O)(=O)C(F)(F)F)ccc3c2C(=O)c2ccc(OCCN3CCCCC3)cc2)cc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP3 O14638 7/20 0.78
ESR1 P03372 9/20 0.75
STS P08842 3/20 0.75
ENPP1 P22413 6/20 0.74
ESR2 Q92731 7/20 0.69
ABCC1 P33527 1/20 0.65
MEN1 O00255 1/20 0.65
PLD2 O14939 1/20 0.65
KDM1A O60341 1/20 0.65
NR1I2 O75469 1/20 0.65
USP2 O75604 1/20 0.65
ALDH1A1 P00352 1/20 0.65
C5 P01031 1/20 0.65
LMNA P02545 1/20 0.65
TP53 P04637 1/20 0.65
FYN P06241 1/20 0.65
PGR P06401 1/20 0.65
CYP3A4 P08684 1/20 0.65
ADRA2A P08913 1/20 0.65
ADORA3 P0DMS8 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18872885 0.96 ESR1 (0.81) ENPP3ESR1STSENPP1ESR2
SCHEMBL1439001 0.94 ENPP3 (0.87) ENPP3ESR1STSENPP1ESR2
SCHEMBL10827879 0.94 ENPP3 (0.87) ENPP3ESR1STSENPP1ESR2
Hydrochloric Acid SCHEMBL1438899 0.94 ENPP3 (0.85) ENPP3ESR1STSENPP1ESR2
SCHEMBL10827744 0.93 ENPP3 (0.85) ENPP3ESR1STSENPP1ESR2
SCHEMBL8596738 0.91 ENPP3 (0.79) ENPP3ESR1STSENPP1ESR2
SCHEMBL5686648 0.89 ENPP3 (0.69) ENPP3ESR1STSENPP1ESR2
SCHEMBL4608181 0.89 STS (0.84) ENPP3ESR1STSESR2ABCC1
SCHEMBL10828093 0.86 ENPP3 (0.73) ENPP3ESR1STSENPP1ESR2
SCHEMBL10827833 0.85 ENPP3 (0.85) ENPP3ESR1STSENPP1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6756388-B1 HAVING PIPERIDINYL AND PHENOLIC FUNCTIONALITY; BONE LOSS; BREAST OR PROSTATE CANCER PFIZER INC. 2004-06-29 US disclosed
EP-0723537-A1 BENZOTHIOPHENES AND RELATED COMPOUNDS AS ESTROGEN AGONISTS PFIZER INC. (US) 1996-07-31 EP disclosed
WO-1995010513-A1 BENZOTHIOPHENES AND RELATED COMPOUNDS AS ESTROGEN AGONISTS PFIZER INC. (US) 1995-04-20 WO disclosed