SCHEMBL6837347

SCHEMBL6837347

CCOC(=O)/C(C)=N\N(Cc1c(Cl)cccc1OCC)C(=O)CC(=O)OC

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
POLB P06746 2/20 0.38
MAPT P10636 3/20 0.36
RORC P51449 1/20 0.35
NLRP3 Q96P20 1/20 0.34
GPR35 Q9HC97 1/20 0.34
CASP1 P29466 1/20 0.34
GAA P10253 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TP53 P04637 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6837376 0.76 ALDH1A1 (0.43) ALDH1A1POLBMAPTRORCNLRP3
SCHEMBL3847139 0.72 ALDH1A1 (0.43) ALDH1A1POLBSMN1; SMN2NPSR1
SCHEMBL3847137 0.72 ALDH1A1 (0.43) ALDH1A1POLBSMN1; SMN2NPSR1
SCHEMBL13873152 0.70 KMT2A (0.44) ALDH1A1POLBMAPTGAASMN1; SMN2
SCHEMBL6837449 0.67 ALDH1A1 (0.47) ALDH1A1POLBMAPTRORC
SCHEMBL3021786 0.65 KMT2A (0.47) ALDH1A1POLBMAPTGAASMN1; SMN2
SCHEMBL393212 0.65 MAPT (0.46) ALDH1A1MAPTGAASMN1; SMN2NPSR1
SCHEMBL393211 0.65 MAPT (0.46) ALDH1A1MAPTGAASMN1; SMN2NPSR1
SCHEMBL3014458 0.63 AKR1B1 (0.41) ALDH1A1MAPTSMN1; SMN2
SCHEMBL14088341 0.63 ALDH1A1 (0.41) ALDH1A1POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
US-7812038-B2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS, INC. (US) 2010-10-12 US disclosed
US-7812038-B2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS, INC. (US) 2010-10-12 US disclosed