SCHEMBL6840529

SCHEMBL6840529

Cc1cccc(-c2ccncn2)c1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.51
MAPK14 Q16539 2/20 0.50
GRM5 P41594 1/20 0.49
BCHE P06276 1/20 0.46
ACHE P22303 1/20 0.46
IDO1 P14902 1/20 0.46
METAP2 P50579 1/20 0.46
KDM1A O60341 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
CYP2D6 P10635 1/20 0.42
CYP2A6 P11509 1/20 0.42
NPY5R Q15761 1/20 0.42
ABL1 P00519 1/20 0.41
BCR P11274 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27663024 0.82 CYP2D6 (0.46) MAPK14GRM5NPC1RAB9ACYP2D6
SCHEMBL29462011 0.80 KMO (0.67) KMOBCHEACHEIDO1METAP2
SCHEMBL2126795 0.80 KMO (0.67) KMOBCHEACHEIDO1METAP2
SCHEMBL14425914 0.79 GRM5 (0.50) KMOMAPK14GRM5CYP2D6
SCHEMBL14425577 0.79 KMO (0.51) KMOMAPK14GRM5CYP2D6
SCHEMBL21742566 0.78 GRM5 (0.43) MAPK14GRM5CYP2D6
SCHEMBL5444466 0.78 MAPK14 (0.45) KMOMAPK14IDO1METAP2
SCHEMBL14519516 0.78 EGFR (0.63) MAPK14IDO1METAP2
SCHEMBL7672405 0.78 GRM5 (0.49) MAPK14GRM5IDO1METAP2NPC1
SCHEMBL20566349 0.78 HSD17B1 (0.58) GRM5METAP2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3503240-A1 ORGANIC SEMICONDUCTOR LAYER Novaled GmbH (DE) 2019-06-26 EP disclosed
US-9716233-B2 Electronic device including a fluoranthene derivative E I DU PONT DE NEMOURS AND COMPANY (US) 2017-07-25 US disclosed
CN-104650117-A Organic compound and application thereof in organic electroluminescence devices BEIJING ETERNAL MATERIAL TECHNOLOGY CO LTD 2015-05-27 CN disclosed
US-8653141-B2 HIV protease inhibiting compounds ABBVIE INC. (US) 2014-02-18 US disclosed
US-20130023463-A1 HIV PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 2013-01-24 US disclosed
US-8193227-B2 HIV protease inhibiting compounds ABBOTT LABORATORIES (US) 2012-06-05 US disclosed
US-20110003827-A1 HIV protease inhibiting compounds ABBVIE INC. 2011-01-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110003827-A1 HIV protease inhibiting compounds SERPINB1, HPN, DNPEP KMO 3581/4885MAPK14 1962/4885GRM5 3144/4885
US-20130023463-A1 HIV PROTEASE INHIBITING COMPOUNDS SERPINB1, HPN, DNPEP KMO 3581/4885MAPK14 1962/4885GRM5 3144/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.