SCHEMBL6842022

SCHEMBL6842022

NC(=O)c1c(-c2ccccc2)cccc1-c1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 2/20 0.63
FOLH1 Q04609 1/20 0.49
FGFR1 P11362 1/20 0.48
SRC P12931 1/20 0.48
FGFR2 P21802 1/20 0.48
FGFR4 P22455 1/20 0.48
FGFR3 P22607 1/20 0.48
CRHBP P24387 1/20 0.48
CRHR2 Q13324 1/20 0.48
HNF4A P41235 1/20 0.48
KMT2A Q03164 3/20 0.47
HSD17B10 Q99714 3/20 0.46
CYP3A4 P08684 2/20 0.46
POLB P06746 1/20 0.46
PARP1 P09874 1/20 0.46
MAPT P10636 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46
RECQL P46063 1/20 0.46
BLM P54132 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1250167 0.88 BCAT2 (0.55) BCAT2FOLH1FGFR1SRCFGFR2
SCHEMBL975812 0.88 BCAT2 (0.55) BCAT2FOLH1FGFR1SRCFGFR2
SCHEMBL901580 0.88 BCAT2 (0.71) BCAT2FOLH1FGFR1SRCFGFR2
SCHEMBL29916354 0.86 BCAT2 (0.63) BCAT2FOLH1FGFR1SRCFGFR2
SCHEMBL30463470 0.86 BCAT2 (0.53) BCAT2FOLH1FGFR1SRCFGFR2
SCHEMBL26554906 0.86 BCAT2 (0.53) BCAT2FOLH1FGFR1SRCFGFR2
SCHEMBL8572487 0.86 BCAT2 (0.53) BCAT2FOLH1FGFR1SRCFGFR2
SCHEMBL570758 0.86 BCAT2 (0.63) BCAT2FOLH1FGFR1SRCFGFR2
SCHEMBL7085409 0.86 BCAT2 (0.53) BCAT2FOLH1FGFR1SRCFGFR2
SCHEMBL30728845 0.86 BCAT2 (0.53) BCAT2FOLH1FGFR1SRCFGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117342955-A Method for preparing 4' -methyl-biphenyl-2-amine 盐城师范学院 2024-01-05 CN claimed
CN-116888112-A Lactams as CBL-B inhibitors 基因泰克公司 2023-10-13 CN disclosed
CN-116848106-A Amides as CBL-B inhibitors 基因泰克公司 2023-10-03 CN disclosed
US-6696380-B2 Procatalysts, catalyst systems, and use in olefin polymerization WESTLAKE LONGVIEW CORPORATION 2004-02-24 US disclosed
US-6677410-B2 COORDINATION CATALYSTS EASTMAN CHEMICAL COMPANY 2004-01-13 US disclosed
US-20030004285-A1 Procatalysts, catalyst systems, and use in olefin polymerization WESTLAKE LONGVIEW CORPORATION 2003-01-02 US disclosed
US-6465383-B2 COORDINATION CATALYST EASTMAN CHEMICAL COMPANY 2002-10-15 US disclosed
US-20010051587-A1 Procatalysts, catalyst systems, and use in olefin polymerization WESTLAKE LONGVIEW CORPORATION 2001-12-13 US disclosed
US-20010031841-A1 Procatalysts, catalyst systems, and use in olefin polymerization WESTLAKE LONGVIEW CORPORATION 2001-10-18 US disclosed
US-20010029286-A1 Procatalysts, catalyst systems, and use in OLEFIN polymerization EASTMAN CHEMICAL COMPANY, A CORP. OF DELAWARE 2001-10-11 US disclosed
US-20010025005-A1 Procatalysts, catalyst systems, and use in olefin polymerization EASTMAN CHEMICAL COMPANY, A CORPORATION OF DELAWARE 2001-09-27 US disclosed
WO-2001051526-A1 PROCATALYSTS COMPRISING BIDENTATE LIGANDS, CATALYST SYSTEMS, AND USE IN OLEFIN POLYMERIZATION EASTMAN CHEMICAL COMPANY (US) 2001-07-19 WO disclosed
WO-2001051527-A1 PROCATALYSTS, CATALYST SYSTEMS, AND USE IN OLEFIN POLYMERIZATION EASTMAN CHEMICAL COMPANY (US) 2001-07-19 WO disclosed
WO-2001051529-A1 PROCATALYSTS COMPRISING BIDENTATE LIGANDS, CATALYST SYSTEMS, AND USE IN OLEFIN POLYMERIZATION EASTMAN CHEMICAL COMPANY (US) 2001-07-19 WO disclosed
WO-2001051528-A1 PROCATALYSTS COMPRISING BIDENTATE LIGANDS, CATALYST SYSTEMS, AND USE IN OLEFIN POLYMERIZATION EASTMAN CHEMICAL COMPANY (US) 2001-07-19 WO disclosed