SCHEMBL6848181

SCHEMBL6848181

OC/C=C/c1ccc(-c2cncnc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
CYP3A4 P08684 1/20 0.43
RECQL P46063 1/20 0.43
ATM Q13315 1/20 0.42
HDAC1 Q13547 4/20 0.42
HDAC2 Q92769 3/20 0.42
HDAC3 O15379 2/20 0.42
KDM1A O60341 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
ERN1 O75460 2/20 0.38
XDH P47989 1/20 0.36
CYP2A6 P11509 1/20 0.35
HDAC4 P56524 2/20 0.35
FLT3 P36888 1/20 0.35
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
GRK6 P43250 1/20 0.33
GRM2 Q14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6848185 1.00 ALDH1A1 (0.43) ALDH1A1CYP3A4RECQLATMHDAC1
SCHEMBL6852489 0.81 CYP17A1 (0.47) ALDH1A1CYP3A4RECQLHDAC1HDAC2
SCHEMBL6852499 0.81 CYP17A1 (0.47) ALDH1A1CYP3A4RECQLHDAC1HDAC2
SCHEMBL6848095 0.81 MKNK1 (0.57) ALDH1A1CYP3A4HDAC1HDAC2HDAC3
SCHEMBL6848092 0.81 MKNK1 (0.57) ALDH1A1CYP3A4HDAC1HDAC2HDAC3
SCHEMBL9276381 0.77 ALDH1A1 (0.62) ALDH1A1CYP3A4RECQLKDM1AHDAC6
SCHEMBL9276383 0.77 ALDH1A1 (0.62) ALDH1A1CYP3A4RECQLKDM1AHDAC6
SCHEMBL14984804 0.76 ALDH1A1 (0.53) ALDH1A1CYP3A4RECQLHDAC1HDAC2
SCHEMBL5580490 0.76 MGLL (0.53) ALDH1A1CYP3A4RECQLHDAC1HDAC2
SCHEMBL5580493 0.76 MGLL (0.53) ALDH1A1CYP3A4RECQLHDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed
EP-1453847-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-09-08 EP disclosed
WO-2003050132-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2003-06-19 WO disclosed