SCHEMBL6848383

SCHEMBL6848383

CCOC(=O)c1ccc(CBr)s1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.55
HDAC4 P56524 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
ALDH1A1 P00352 5/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
CDC7 O00311 1/20 0.43
DBF4 Q9UBU7 1/20 0.43
TSHR P16473 2/20 0.43
PLK1 P53350 1/20 0.42
CYP4F2 P78329 1/20 0.42
CYP4A11 Q02928 1/20 0.42
GAA P10253 3/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 4/20 0.41
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12838390 0.86 HDAC3 (0.58) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL2653117 0.84 HDAC3 (0.57) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL15888182 0.84 TSHR (0.49) ALDH1A1SMN1; SMN2TSHRMAPTHPGD
SCHEMBL8010507 0.83 ALDH1A1 (0.39) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL7018973 0.83 HDAC3 (0.73) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL6814615 0.83 HDAC3 (0.55) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL348559 0.82 LMNA (0.51) ALDH1A1SMN1; SMN2TSHRMAPTHPGD
SCHEMBL2653067 0.82 HDAC3 (0.51) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL2653869 0.81 HDAC3 (0.54) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL1731610 0.81 ALDH1A1 (0.38) HDAC3HDAC4HDAC1HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119390668-A Compound with ketoxime ether structure and application thereof 复旦大学 2025-02-07 CN disclosed
CN-115368306-B HDAC inhibitor containing tetrahydroisoquinoline structure, composition and application thereof 安徽中医药大学 2023-12-22 CN disclosed
CN-110234656-B Exonucleotidase inhibitors and methods of use thereof 卡利泰拉生物科技公司 2023-02-28 CN disclosed
US-20230002437-A1 ECTONUCLEOTIDASE INHIBITORS AND METHODS OF USE THEREOF ANTENGENE THERAPEUTICS LIMITED (CN) 2023-01-05 US disclosed
CN-115368306-A HDAC (Histone deacetylase) inhibitor containing tetrahydroisoquinoline structure, composition and application thereof 安徽中医药大学 2022-11-22 CN disclosed
US-11208414-B2 Ectonucleotidase inhibitors and methods of use thereof CALITHERA BIOSCIENCES, INC. (US) 2021-12-28 US disclosed
US-11174261-B2 2021-11-16 US disclosed
US-11034715-B2 Ectonucleotidase inhibitors and methods of use thereof CALITHERA BIOSCIENCES, INC. (US) 2021-06-15 US disclosed
US-20200223882-A1 Ectonucleotidase Inhibitors and Methods of Use Thereof ANTENGENE THERAPEUTICS LIMITED (CN) 2020-07-16 US disclosed
US-20200087310-A1 Ectonucleotidase Inhibitors and Methods of Use Thereof ANTENGENE THERAPEUTICS LIMITED (CN) 2020-03-19 US disclosed
EP-0861843-B1 Fluorescent ionophoric compounds with a cryptand/crown-ether portion and a coumarin portion, their preparation and their use for measuring metal cation concentrations TERUMO CARDIOVASCULAR SYS (US) 2004-07-14 EP disclosed
US-6624188-B1 Administered to treat or prevent one or more of the diseases and conditions selected from the group consisting of dermatoses, atherosclerosis and restenosis resulting from neointimal hyperproliferation, non-malignant and ALLERGAN, INC. 2003-09-23 US disclosed
US-5958782-A FLUORESCENT IONOPHORIC COMPOUND IS DISCLOSED THAT INCLUDES A COMPLEXING MOIETY, SUCH AS A CRYPTAND OR CROWN-ETHER PORTION, AND A FLUORESCING MOIETY SUCH AS A COUMARIN PORTION MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1999-09-28 US disclosed
EP-0861843-A2 Fluorescent ionophoric compounds with a cryptand/crown-ether portion and a coumarin portion, their preparation and their use for measuring metal cation concentrations MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1998-09-02 EP disclosed
US-5434173-A Administering to treat acne, psoriasis, eczema, dermatitis, and other skin disorders ALLERGAN, INC. (US) 1995-07-18 US disclosed
US-5391753-A Tumor inhibiting agents; useful for treating dermatological conditions and rheumatic illnesses ALLERGAN, INC. (US) 1995-02-21 US disclosed
EP-0626955-A1 HETEROARYL SUBSTITUTED PHENYLETHENYL COMPOUNDS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 1994-12-07 EP disclosed
US-5324840-A Skin disorders ALLERGAN, INC. (US) 1994-06-28 US disclosed
WO-1993016067-A1 HETEROARYL SUBSTITUTED PHENYLETHENYL COMPOUNDS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 1993-08-19 WO disclosed
US-4273782-A FOR USE IN CARDIOVASCULAR DISORDERS AND COMPLICATIONS OF DIABETES PFIZER INC. (US) 1981-06-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200223882-A1 Ectonucleotidase Inhibitors and Methods of Use Thereof NT5E, ENTPD5, NT5C2 HDAC3 1985/4885HDAC4 2614/4885HDAC1 3062/4885
US-11034715-B2 Ectonucleotidase inhibitors and methods of use thereof NT5E, ENTPD5, NT5C2 HDAC3 1985/4885HDAC4 2614/4885HDAC1 3062/4885
US-11174261-B2 ENTPD5, NT5E, ENTPD1 HDAC3 1238/4885HDAC4 1841/4885HDAC1 2180/4885
US-11208414-B2 Ectonucleotidase inhibitors and methods of use thereof ENTPD5, NT5E, ENTPD1 HDAC3 1929/4885HDAC4 2651/4885HDAC1 2814/4885
US-20200087310-A1 Ectonucleotidase Inhibitors and Methods of Use Thereof NT5E, ENTPD5, NT5C2 HDAC3 1985/4885HDAC4 2614/4885HDAC1 3062/4885
US-20230002437-A1 ECTONUCLEOTIDASE INHIBITORS AND METHODS OF USE THEREOF NT5E, ENTPD5, NT5C2 HDAC3 1985/4885HDAC4 2614/4885HDAC1 3062/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.