SCHEMBL6850299

SCHEMBL6850299

O=C(O)N1CCc2c(n3c4c(cccc24)CCC3Cc2ccccc2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
TDP1 Q9NUW8 1/20 0.36
PTGDR2 Q9Y5Y4 3/20 0.36
CDK4 P11802 2/20 0.36
CCND1 P24385 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
FABP4 P15090 3/20 0.35
FABP3 P05413 1/20 0.35
MTNR1A P48039 2/20 0.35
MTNR1B P49286 1/20 0.35
CCNE2 O96020 1/20 0.35
PRKACA P17612 1/20 0.35
PRKACG P22612 1/20 0.35
PRKACB P22694 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
GRIN2B Q13224 1/20 0.35
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6491761 0.82 CHRM1 (0.38) PTGDR2HTR2B
SCHEMBL7037197 0.74 DPP4 (0.35) PTGDR2MEN1KMT2AFABP4FABP3
SCHEMBL6496231 0.74 SMN1; SMN2 (0.50) PTGDR2MEN1KMT2AGRIN2BCYP2C19
SCHEMBL6851617 0.73 PTGDR2 (0.34) PTGDR2MEN1KMT2AFABP4FABP3
SCHEMBL6851622 0.73 LTB4R (0.37) PTGDR2MEN1KMT2ACYP2C9
SCHEMBL6847665 0.72 PTGDR2 (0.33) PTGDR2MEN1KMT2AFABP4FABP3
SCHEMBL7030588 0.72 MCL1 (0.52) KDM4ETDP1MEN1KMT2ACYP2C9
SCHEMBL6485143 0.68 HTR2C (0.46) KDM4ETDP1PTGDR2MEN1KMT2A
SCHEMBL6496372 0.66 PTGDR2 (0.36) KDM4ETDP1PTGDR2MEN1KMT2A
SCHEMBL17634168 0.65 ALDH1A1 (0.40) KDM4ECDK4CCND1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173440-B1 TETRACYCLIC AZEPINOINDOLE COMPOUNDS AS 5-HT RECEPTOR LIGANDS UPJOHN CO (US) 2004-09-15 EP claimed