Bromide

Bromide

SCHEMBL6851089

Br.Cn1c(=O)oc2cccc(C(C)(C)C)c21

nearest known ligand 0.34

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.34
ALDH1A1 P00352 3/20 0.33
HPGD P15428 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PRKDC P78527 1/20 0.32
TSHR P16473 2/20 0.32
MAPK1 P28482 2/20 0.32
USP2 O75604 1/20 0.32
CYP1A2 P05177 1/20 0.31
GLA P06280 1/20 0.31
LMNA P02545 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PKM P14618 3/20 0.31
GABRA1 P14867 1/20 0.31
GABRB2 P47870 1/20 0.31
POLB P06746 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25536906 0.98 CA2 (0.35) CA2ALDH1A1HPGDNPSR1PRKDC
SCHEMBL3354467 0.75 POLB (0.41) ALDH1A1HPGDNPSR1TSHRMAPK1
SCHEMBL5541190 0.74 ALDH1A1 (0.41) ALDH1A1HPGDNPSR1TSHRMAPK1
SCHEMBL5537338 0.74 JAK2 (0.39) ALDH1A1HPGDNPSR1TSHRMAPK1
SCHEMBL5543644 0.74 MEN1 (0.38) ALDH1A1HPGDNPSR1TSHRMAPK1
SCHEMBL14199897 0.71 TSHR (0.37) CA2ALDH1A1HPGDNPSR1TSHR
SCHEMBL24656305 0.71 HTR1A (0.38) CA2ALDH1A1HPGDNPSR1PRKDC
SCHEMBL3552088 0.69 ALDH1A1 (0.38) ALDH1A1HPGDMAPK1CYP1A2LMNA
SCHEMBL20650931 0.66 CA2 (0.44) CA2ALDH1A1NPSR1TSHRCYP1A2
SCHEMBL637681 0.66 PTPN1 (0.41) ALDH1A1HPGDMAPK1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1394152-A1 2-IMINOIMIDAZOLE DERIVATIVES (1) Eisai Co., Ltd. (JP) 2004-03-03 EP disclosed