SCHEMBL6852633

SCHEMBL6852633

OC/C=C/c1ccc2cccnc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
CASP1 P29466 1/20 0.50
CASP7 P55210 1/20 0.50
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
CYP3A4 P08684 5/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6852642 1.00 ALDH1A1 (0.50) ALDH1A1MEN1KMT2ACASP1CASP7
SCHEMBL3149307 0.87 NPC1 (0.60) ALDH1A1MEN1KMT2ACASP1HDAC3
SCHEMBL4105395 0.87 NPC1 (0.60) ALDH1A1MEN1KMT2ACASP1HDAC3
SCHEMBL5800253 0.81 MAPT (0.47) ALDH1A1MEN1KMT2ACASP1CASP7
SCHEMBL5800255 0.81 MAPT (0.47) ALDH1A1MEN1KMT2ACASP1CASP7
SCHEMBL12132425 0.80 ALDH1A1 (0.46) ALDH1A1MEN1KMT2ACASP1CASP7
SCHEMBL9970465 0.80 NPC1 (0.54) ALDH1A1MEN1KMT2ACASP1CASP7
SCHEMBL6851745 0.80 CYP3A4 (0.52) ALDH1A1MEN1KMT2ACYP3A4RECQL
SCHEMBL6851757 0.80 CYP3A4 (0.52) ALDH1A1MEN1KMT2ACYP3A4RECQL
SCHEMBL6656717 0.78 ALDH1A1 (0.50) ALDH1A1MEN1KMT2ACASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed
EP-1453847-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-09-08 EP disclosed
WO-2003050132-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2003-06-19 WO disclosed