SCHEMBL12132425

SCHEMBL12132425

CC(C)C/C=C/c1ccc2cccnc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
HTT P42858 1/20 0.46
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
NR4A2 P43354 1/20 0.42
NPC1 O15118 2/20 0.42
MAPT P10636 2/20 0.42
RAB9A P51151 2/20 0.42
CASP3 P42574 1/20 0.42
ATM Q13315 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12132427 0.88 NPC1 (0.56) ALDH1A1HTTMEN1KMT2ACASP1
SCHEMBL12132442 0.81 CYP3A4 (0.42) ALDH1A1MEN1KMT2ACASP1CASP7
SCHEMBL13723845 0.81 CHRNB2 (0.41) KMT2ARAB9AOGACHRNB2CHRNA4
SCHEMBL6852642 0.80 ALDH1A1 (0.50) ALDH1A1CYP1A2CYP2C19HTTMEN1
SCHEMBL6852633 0.80 ALDH1A1 (0.50) ALDH1A1CYP1A2CYP2C19HTTMEN1
SCHEMBL5800255 0.78 MAPT (0.47) ALDH1A1CYP1A2CYP2C19HTTMEN1
SCHEMBL5800253 0.78 MAPT (0.47) ALDH1A1CYP1A2CYP2C19HTTMEN1
SCHEMBL13722897 0.77 CHRNB2 (0.40) MEN1KMT2ANPC1MAPTRAB9A
SCHEMBL9970465 0.76 NPC1 (0.54) ALDH1A1CYP1A2CYP2C19HTTMEN1
SCHEMBL5620728 0.76 HTT (0.60) ALDH1A1CYP1A2CYP2C19HTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063021-B2 Ketolide anti-infective compounds KOSAN BIOSCIENCES INCORPORATED (US) 2011-11-22 US disclosed
US-8063021-B2 Ketolide anti-infective compounds KOSAN BIOSCIENCES INCORPORATED (US) 2011-11-22 US disclosed