SCHEMBL6853783

SCHEMBL6853783

COc1cc(Cn2c(=O)c3cc(Br)ccc3n3c(N4CCCC4)nnc23)cc(OC)c1OC

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
HPGD P15428 1/20 0.37
HSP90AA1 P07900 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
POLB P06746 1/20 0.37
LMNA P02545 2/20 0.37
TSHR P16473 1/20 0.37
MAPT P10636 3/20 0.37
TP53 P04637 3/20 0.37
USP2 O75604 1/20 0.36
THRB P10828 1/20 0.36
KDM4E B2RXH2 1/20 0.35
PDE5A O76074 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6854057 0.91 MAPT (0.42) ALDH1A1HPGDHSP90AA1NPSR1LMNA
SCHEMBL6854129 0.90 MAPT (0.41) ALDH1A1HPGDHSP90AA1NPSR1LMNA
SCHEMBL6855972 0.90 MAPT (0.41) ALDH1A1HPGDHSP90AA1NPSR1LMNA
SCHEMBL6850259 0.89 MAPT (0.41) ALDH1A1HPGDHSP90AA1NPSR1LMNA
SCHEMBL6854048 0.87 PIK3R1 (0.46) ALDH1A1HSP90AA1NPSR1MAPTTP53
SCHEMBL6854439 0.84 MAPT (0.51) ALDH1A1HPGDNPSR1LMNATSHR
SCHEMBL6850125 0.84 L3MBTL1 (0.48) ALDH1A1LMNATSHRMAPTTP53
SCHEMBL7146999 0.84 PIK3R1 (0.40) ALDH1A1HPGDLMNATSHRMAPT
SCHEMBL7529993 0.84 PIK3R1 (0.40) ALDH1A1HPGDLMNATSHRMAPT
SCHEMBL6854145 0.83 L3MBTL1 (0.47) ALDH1A1HPGDLMNATSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6828315-B1 Anti- inflammatories, anti-allergics, bronchodilatators, anti-asthmatics, or TNF alpha inhibitors WARNER-LAMBERT LLC 2004-12-07 US claimed
US-6828315-B1 Anti- inflammatories, anti-allergics, bronchodilatators, anti-asthmatics, or TNF alpha inhibitors WARNER-LAMBERT LLC 2004-12-07 US disclosed
EP-1177195-B1 1-AMINO TRIAZOLO 4,3-a! QUINAZOLINE-5-ONES AND OR -5-THIONES INHIBITING PHOSPHODIESTERASE IV WARNER LAMBERT CO (US) 2003-03-19 EP disclosed