SCHEMBL6854844

SCHEMBL6854844

O=c1[nH]c2nnc(N3CCCCCC3)n2c2ccc(Cl)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAT2A P31153 2/20 0.43
PDE10A Q9Y233 1/20 0.39
HRH4 Q9H3N8 2/20 0.39
HTR3A P46098 1/20 0.39
NPC1 O15118 2/20 0.38
HPGD P15428 2/20 0.38
TSHR P16473 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 1/20 0.38
NFKB1 P19838 1/20 0.38
GFER P55789 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
MAP2K7 O14733 1/20 0.37
PIM1 P11309 1/20 0.36
PIM2 Q9P1W9 1/20 0.36
ALDH1A1 P00352 2/20 0.36
HSD17B10 Q99714 2/20 0.36
CHKA P35790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6855823 0.84 PIM1 (0.35) NPC1RAB9APIM1PIM2ALDH1A1
SCHEMBL6858242 0.82 HPGD (0.41) HPGDTSHRSMN1; SMN2GFERALDH1A1
SCHEMBL6858355 0.80 ALDH1A1 (0.33) HPGDTSHRRAB9ASMN1; SMN2ALDH1A1
SCHEMBL6855784 0.75 MAPT (0.46) MAT2AHRH4HTR3AHPGDTSHR
SCHEMBL6850076 0.75 MAPT (0.46) MAT2AHRH4HTR3AHPGDTSHR
SCHEMBL6854165 0.75 MAPT (0.46) MAT2AHRH4HTR3AHPGDTSHR
SCHEMBL6855846 0.73 MAPT (0.46) HRH4HTR3AHPGDTSHRSMN1; SMN2
SCHEMBL6850089 0.72 PLK1 (0.44) HPGDTP53ALDH1A1HSD17B10LMNA
SCHEMBL6858251 0.71 ALDH1A1 (0.50) MAT2AHPGDTSHRSMN1; SMN2ALDH1A1
SCHEMBL6853905 0.71 L3MBTL1 (0.47) TP53ALDH1A1LMNAPOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6828315-B1 Anti- inflammatories, anti-allergics, bronchodilatators, anti-asthmatics, or TNF alpha inhibitors WARNER-LAMBERT LLC 2004-12-07 US disclosed
EP-1177195-B1 1-AMINO TRIAZOLO 4,3-a! QUINAZOLINE-5-ONES AND OR -5-THIONES INHIBITING PHOSPHODIESTERASE IV WARNER LAMBERT CO (US) 2003-03-19 EP disclosed