SCHEMBL6856480

SCHEMBL6856480

O=C(O)c1c[nH]nc1Cc1cccc(F)c1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 3/20 0.54
NR4A2 P43354 2/20 0.44
BRS3 P32247 1/20 0.43
KDM5A P29375 1/20 0.42
KDM4C Q9H3R0 1/20 0.42
KDM5B Q9UGL1 1/20 0.42
PDE10A Q9Y233 1/20 0.40
DAO P14920 1/20 0.40
PARP1 P09874 1/20 0.39
SLC1A1 P43005 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1697133 0.84 NR4A2 (0.48) NR4A2DAO
SCHEMBL4017043 0.84 HCAR2 (0.45) HCAR2KDM5AKDM4CKDM5BPARP1
SCHEMBL5779014 0.83 PDE3B (0.49) HCAR2
SCHEMBL15622305 0.74 AR (0.47) BRS3KDM5AKDM4CKDM5B
SCHEMBL28105342 0.74 HCAR2 (0.52) HCAR2NR4A2BRS3SLC1A1
SCHEMBL22534331 0.73 KDM5B (0.46) BRS3KDM5AKDM4CKDM5BPARP1
SCHEMBL9937529 0.73 HCAR2 (0.51) HCAR2NR4A2BRS3SLC1A1
SCHEMBL4448337 0.73 BRS3 (0.47) HCAR2NR4A2BRS3KDM5AKDM4C
SCHEMBL28214966 0.72 DCLRE1B (0.47) NR4A2
SCHEMBL28117926 0.72 TSHR (0.57) HCAR2NR4A2BRS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444233-A2 A 2B? ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS, INC. (US) 2004-08-11 EP claimed
WO-2003042214-A2 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS, INC. (US) 2003-05-22 WO claimed