SCHEMBL6856979

SCHEMBL6856979

CCC(CC)N1CCc2ccc(CNC(=O)c3cnc(N(C)C[C@H](C)OC)nc3)cc2CC1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TP53 P04637 6/20 0.39
THRB P10828 2/20 0.39
PRKAB2 O43741 1/20 0.38
PRKAG1 P54619 1/20 0.38
PRKAA2 P54646 1/20 0.38
PRKAA1 Q13131 1/20 0.38
PRKAG3 Q9UGI9 1/20 0.38
PRKAG2 Q9UGJ0 1/20 0.38
PRKAB1 Q9Y478 1/20 0.38
LMNA P02545 7/20 0.37
POLB P06746 3/20 0.37
MAPK14 Q16539 1/20 0.36
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2191319 0.85 HRH3 (0.48) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL2191302 0.85 HRH3 (0.48) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL2266798 0.78 HRH3 (0.51) TP53THRBPRKAB2PRKAG1PRKAA2
SCHEMBL2267296 0.78 HRH3 (0.51) TP53THRBPRKAB2PRKAG1PRKAA2
SCHEMBL2269194 0.71 HRH3 (0.49) LMNAPOLB
SCHEMBL2223911 0.71 HRH3 (0.49) LMNAPOLB
SCHEMBL1787185 0.70 PRKAB2 (0.42) TP53THRBPRKAB2PRKAG1PRKAA2
SCHEMBL1787184 0.70 HRH3 (0.51) TP53THRBPRKAB2PRKAG1PRKAA2
SCHEMBL1789991 0.68 HRH3 (0.51) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL1789988 0.68 HRH3 (0.51) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011083314-A1 BENZAZEPINE DERIVATIVES FOR THE TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 WO disclosed