SCHEMBL6857308

SCHEMBL6857308

CC(=O)c1ccccc1NC(=O)C(=O)Nc1ccccc1C(C)=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.57
RAB9A P51151 4/20 0.57
PDK1 Q15118 1/20 0.57
PDK2 Q15119 1/20 0.57
PDK3 Q15120 1/20 0.57
PDK4 Q16654 1/20 0.57
CNR2 P34972 1/20 0.54
CYP2C19 P33261 3/20 0.53
POLB P06746 1/20 0.53
DHODH Q02127 1/20 0.53
TRPM8 Q7Z2W7 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.51
KDM4E B2RXH2 2/20 0.49
LMNA P02545 1/20 0.49
AKR1C3 P42330 1/20 0.49
AKR1C2 P52895 1/20 0.49
KMT2A Q03164 1/20 0.47
ALDH1A1 P00352 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
HPGD P15428 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6855309 0.94 PDK1 (0.53) NPC1RAB9APDK1PDK2PDK3
SCHEMBL14397793 0.90 CYP2C19 (0.58) NPC1RAB9APDK1PDK2PDK3
SCHEMBL505353 0.87 CYP2C19 (0.69) NPC1RAB9APDK1PDK2PDK3
SCHEMBL29808973 0.87 CYP2C19 (0.69) NPC1RAB9APDK1PDK2PDK3
SCHEMBL18415571 0.87 ALDH1A1 (0.50) NPC1RAB9APDK1PDK2PDK3
SCHEMBL2943260 0.85 PDK1 (0.56) NPC1RAB9APDK1PDK2PDK3
SCHEMBL2837597 0.85 POLB (0.56) NPC1RAB9APDK1PDK2PDK3
SCHEMBL27644581 0.85 PDK1 (0.56) NPC1RAB9APDK1PDK2PDK3
SCHEMBL6428947 0.84 PDK1 (0.51) NPC1RAB9APDK1PDK2PDK3
SCHEMBL28879810 0.83 PDK1 (0.54) NPC1RAB9APDK1PDK2PDK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6737193-B2 ACTIVE MATERIALS IN THE POSITIVE ELECTRODES OF BATTERIES. NOVEL METHODS FOR PREPARING THE TETRAKETOPIPERAZINE UNIT-CONTAINING COMPOUNDS INCLUDE: (I) REACTING AN OXALYL HALIDE AND AN OXAMIDE, AND ADDING WATER OR AN AQUEOUS ALKALI IM&T RESEARCH, INC. 2004-05-18 US disclosed
US-20030148188-A1 Active materials in the positive electrodes of batteries. Novel methods for preparing the tetraketopiperazine unit-containing compounds include: (i) reacting an oxalyl halide and an oxamide, and adding water or an aqueous alkali IM&T RESEARCH, INC. 2003-08-07 US disclosed