SCHEMBL6860667

SCHEMBL6860667

O=C(O)c1ccc(Cn2nc(C(F)(F)F)c3c2NCCC3)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.44
TSHR P16473 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MAPT P10636 5/20 0.41
POLB P06746 1/20 0.41
TP53 P04637 2/20 0.41
GAA P10253 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HTT P42858 1/20 0.41
KDM4E B2RXH2 1/20 0.41
RAB9A P51151 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
POLQ O75417 1/20 0.41
CYP1A2 P05177 3/20 0.40
CYP2C9 P11712 2/20 0.40
GRIA2 P42262 2/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
GCGR P47871 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6862396 0.87 POLB (0.45) LMNATSHRNPSR1MAPTPOLB
SCHEMBL6860631 0.86 OPRD1 (0.43) MAPTPOLBPOLQCYP1A2CYP2C9
SCHEMBL13521117 0.82 LMNA (0.62) LMNATSHRNPSR1MAPTPOLB
SCHEMBL6860642 0.81 SMN1; SMN2 (0.49) LMNATSHRMAPTPOLBTP53
SCHEMBL12997897 0.81 GRIA2 (0.53) TSHRMAPTGAAKDM4ECYP1A2
SCHEMBL6860475 0.78 LMNA (0.44) LMNATSHRNPSR1MAPTPOLB
SCHEMBL13521113 0.72 LMNA (0.63) LMNATSHRNPSR1MAPTTP53
SCHEMBL13773366 0.72 MAPT (0.69) LMNATSHRNPSR1MAPTPOLB
SCHEMBL1007029 0.71 LMNA (0.56) LMNATSHRNPSR1MAPTPOLB
SCHEMBL13521108 0.71 LMNA (0.66) LMNATSHRNPSR1MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011036889-A1 HETEROCYCLIC COMPOUND 武田薬品工業株式会社 (JP) 2011-03-31 WO disclosed