SCHEMBL6862756

SCHEMBL6862756

Cc1ncc(C[n+]2csc(CCOP(=O)([O-])OC[C@H]3O[C@@H](n4cnc5c(N)ncnc54)C(O)C3O)c2C)c(N)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.53
P2RY1 P47900 8/20 0.52
P2RY2 P41231 3/20 0.52
P2RY11 Q96G91 3/20 0.52
SRC P12931 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
DNPH1 O43598 1/20 0.52
PRKAB2 O43741 1/20 0.52
TRPM2 O94759 1/20 0.52
LDHA P00338 1/20 0.52
ADRB2 P07550 1/20 0.52
FBP1 P09467 1/20 0.52
ADORA1 P30542 1/20 0.52
PRKAG1 P54619 1/20 0.52
PRKAA2 P54646 1/20 0.52
PDE4D Q08499 1/20 0.52
KCNH2 Q12809 1/20 0.52
PRKAA1 Q13131 1/20 0.52
PDE3A Q14432 1/20 0.52
TAS1R3 Q7RTX0 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31005215 0.93 P2RY1 (0.56) P2RY1P2RY2SRCSMN1; SMN2TRPM2
SCHEMBL14636151 0.91 TKT (0.56) TDP1P2RY1P2RY2P2RY11SRC
SCHEMBL675658 0.90 LMNA (0.58) TDP1P2RY1P2RY2P2RY11SRC
Adenosine SCHEMBL2702312 0.88 LMNA (0.56) TDP1P2RY1P2RY2SRCSMN1; SMN2
Cocarboxylase SCHEMBL14636148 0.86 LMNA (0.63) TDP1P2RY1P2RY2SRCSMN1; SMN2
Adenosine SCHEMBL675657 0.86 LMNA (0.62) TDP1P2RY1P2RY2SRCSMN1; SMN2
Hydrochloric Acid SCHEMBL7793647 0.85 TDP1 (0.55) TDP1LMNATKTRNASEL
Adenosine SCHEMBL6862749 0.84 HSP90AA1 (0.53) TDP1P2RY1P2RY2P2RY11SRC
Adenosine SCHEMBL15347371 0.83 HSP90AA1 (0.57) SMN1; SMN2ADORA1
Adenosine Triphosphate SCHEMBL28087656 0.80 P2RY1 (0.56) P2RY1P2RY2SRCSMN1; SMN2TRPM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1410302-A2 CLASSIFICATION OF POLYPEPTIDES BY LIGAND GEOMETRY AND RELATED METHODS Triad Therapeutics, Inc. (US) 2004-04-21 EP claimed
US-20030236630-A1 Classification of polypeptides by ligand geometry and related methods TRIAD THERAPEUTICS, INC. 2003-12-25 US claimed
US-20020133296-A1 Classification of polypeptides by ligand geometry and related methods TRIAD THERAPEUTICS, INC. 2002-09-19 US claimed
WO-2002056236-A2 CLASSIFICATION OF POLYPEPTIDES BY LIGAND GEOMETRY AND RELATED METHODS TRIAD THERAPEUTICS INC (US) 2002-07-18 WO claimed