SCHEMBL6863347

SCHEMBL6863347

CCOC(=O)C[C@H]1Cc2cc(C#N)c(C(=O)C=O)cc2Cc2ccccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 4/20 0.36
MTNR1B P49286 4/20 0.36
CASR P41180 1/20 0.36
NLRP3 Q96P20 1/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
ALDH1A1 P00352 6/20 0.33
L3MBTL1 Q9Y468 4/20 0.33
ITGB3 P05106 3/20 0.33
ITGAV P06756 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
POLB P06746 1/20 0.33
MAPK1 P28482 1/20 0.33
ITGB1 P05556 1/20 0.33
ITGA2B P08514 1/20 0.33
ITGB5 P18084 1/20 0.33
CYP1A2 P05177 1/20 0.33
KDM4E B2RXH2 4/20 0.33
HSD17B10 Q99714 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6857814 0.89 MTNR1A (0.36) MTNR1AMTNR1BCASRNLRP3LMNA
SCHEMBL6857908 0.86 MTNR1A (0.38) MTNR1AMTNR1BCASRNLRP3LMNA
SCHEMBL6862157 0.86 MTNR1A (0.38) MTNR1AMTNR1BCASRNLRP3LMNA
SCHEMBL6862777 0.76 MTNR1A (0.40) MTNR1AMTNR1BALDH1A1ITGB3ITGAV
SCHEMBL6862775 0.76 MTNR1A (0.40) MTNR1AMTNR1BALDH1A1ITGB3ITGAV
SCHEMBL7516493 0.75 MTNR1A (0.45) MTNR1AMTNR1BITGB3ITGAVITGB1
SCHEMBL6857764 0.75 MTNR1A (0.45) MTNR1AMTNR1BITGB3ITGAVITGB1
SCHEMBL6857996 0.75 MTNR1A (0.45) MTNR1AMTNR1BITGB3ITGAVITGB1
SCHEMBL19984866 0.75 CYP1A2 (0.49) MTNR1AMTNR1BPOLBCYP1A2HSD17B10
SCHEMBL7442839 0.74 SRD5A2 (0.44) MTNR1AMTNR1BITGB3ITGAVITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973730-B1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2004-06-16 EP disclosed
US-6294531-B1 AMINOALKANOLS AS BLOOD COAGULANTS SMITHKLINE BEECHAM CORPORATION 2001-09-25 US disclosed