SCHEMBL6863375

SCHEMBL6863375

c1ccc(-c2cccc(CN3CCN(c4cccc5c4OCN5)CC3)c2)cc1

nearest known ligand 0.80

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 16/20 0.80
HTR1A P08908 13/20 0.80
DRD4 P21917 4/20 0.57
HTR7 P34969 1/20 0.47
DRD3 P35462 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863614 0.79 DRD2 (0.70) DRD2HTR1ADRD4HTR7DRD3
SCHEMBL13533020 0.79 HTR1A (1.00) DRD2HTR1ADRD4HTR7DRD3
SCHEMBL13533014 0.78 DRD2 (0.73) DRD2HTR1ADRD4HTR7DRD3
SCHEMBL15938505 0.78 DRD4 (0.70) DRD2HTR1ADRD4HTR7
SCHEMBL14507216 0.77 HTR1A (0.91) DRD2HTR1ADRD4HTR7DRD3
SCHEMBL15937917 0.76 DRD2 (0.69) DRD2HTR1ADRD4HTR7DRD3
SCHEMBL13533022 0.76 HTR1A (0.71) DRD2HTR1ADRD4HTR7DRD3
SCHEMBL15938316 0.76 DRD4 (0.67) DRD2HTR1ADRD4HTR7
SCHEMBL15937598 0.75 DRD4 (0.67) DRD2HTR1ADRD4DRD3
SCHEMBL7499884 0.75 DRD4 (0.67) DRD2HTR1ADRD4HTR7DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088838-A1 NOVEL 6,6A,7,8,9,10-HEXAHYDRO-4H-4,8,10A-TRIAZA-ACEPHENANTHRYLENE DERIVATIVES AS DOPAMINE D2 LIGANDS H. LUNDBECK A/S (DK) 2011-07-28 WO disclosed