SCHEMBL6863403

SCHEMBL6863403

CCNC(=O)Oc1cc(N)n2nc(-c3nccs3)nc2c1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.36
HPGD P15428 1/20 0.34
ADORA1 P30542 3/20 0.34
CSNK1D P48730 2/20 0.34
ADORA2B P29275 1/20 0.34
KLKB1 P03952 1/20 0.33
HSF1 Q00613 1/20 0.32
KMT2A Q03164 1/20 0.32
SMPD3 Q9NY59 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870768 0.91 BCHE (0.36) HSF1
SCHEMBL6869933 0.84 ADORA2A (0.41) ADORA2AADORA1ADORA2BHSF1KMT2A
SCHEMBL6871432 0.83 ADORA2A (0.40) ADORA2AHPGDADORA1CSNK1DADORA2B
SCHEMBL6869532 0.83 ADORA2A (0.36) ADORA2AADORA1ADORA2BHSF1
SCHEMBL6873153 0.82 ADORA2A (0.38) ADORA2AHPGDADORA1ADORA2BHSF1
SCHEMBL6874251 0.82 ADORA2A (0.43) ADORA2AHPGDADORA1ADORA2BHSF1
SCHEMBL6863200 0.80 ADORA2A (0.38) ADORA2AHPGDADORA1ADORA2BHSF1
SCHEMBL6871963 0.80 ADORA2A (0.35) ADORA2AADORA1ADORA2B
SCHEMBL6867675 0.79 ADORA2A (0.33) ADORA2AADORA1ADORA2B
SCHEMBL6870655 0.78 ADORA2A (0.33) ADORA2AADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP claimed