SCHEMBL6863511

SCHEMBL6863511

Cc1cc(NC(=O)C(=O)O)cc(C)c1Cc1ccc(O)c(Cc2ccc(F)cc2)c1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
THRA P10827 10/20 0.43
THRB P10828 10/20 0.43
OPRK1 P41145 1/20 0.38
EGFR P00533 1/20 0.38
ERBB2 P04626 1/20 0.38
SLC7A5 Q01650 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6862641 0.86 SMN1; SMN2 (0.43) THRATHRBOPRK1
SCHEMBL23983024 0.83 THRA (0.60) THRATHRB
SCHEMBL27702907 0.82 THRA (0.41) THRATHRBOPRK1
SCHEMBL13399172 0.80 THRA (0.45) THRATHRBOPRK1
SCHEMBL3162305 0.78 THRA (0.42) THRATHRBOPRK1
SCHEMBL3162304 0.78 THRA (0.54) THRATHRBOPRK1
SCHEMBL6864350 0.78 THRA (0.63) THRATHRB
SCHEMBL23003762 0.77 THRB (0.66) THRATHRB
SCHEMBL6858246 0.77 SMN1; SMN2 (0.46) OPRK1
SCHEMBL27053517 0.75 MEN1 (0.48) THRATHRBOPRK1SLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1286957-B1 DIPHENYLMETHANE DERIVATIVES BAYER HEALTHCARE AG (DE) 2004-11-03 EP disclosed
US-6803480-B2 THERAPEUTIC TREATMENT AND/OR PROPHYLAXIS OF ARTERIOSCLEROSIS AND HYPERCHOLESTEROLAEMIA BAYER AKTIENGESELLSCHAFT (DE) 2004-10-12 US disclosed
US-20030203898-A1 Therapeutic treatment and/or prophylaxis of arteriosclerosis and hypercholesterolaemia BAYER AKTIENGESELLSCHAFT (DE) 2003-10-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030203898-A1 Therapeutic treatment and/or prophylaxis of arteriosclerosis and hypercholesterolaemia APOB, HMGCR, PCSK9 THRA 2817/4885THRB 2653/4885OPRK1 4591/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.