SCHEMBL686359

SCHEMBL686359

CCC[C@H](O)C(CNCC(C)C)N(C(=O)O)C(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 2/20 0.33
CCR5 P51681 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL686358 1.00 CCR2 (0.33) CCR2CCR5CYP2D6CYP2C19
SCHEMBL14910434 0.81 LMNA (0.35)
SCHEMBL14909876 0.75 CHRM1 (0.34)
SCHEMBL609656 0.72 ANPEP (0.42)
SCHEMBL80781 0.71 CYP2D6 (0.34) CYP2D6CYP2C19
SCHEMBL14909757 0.69 TSHR (0.31)
SCHEMBL4799165 0.68 CCR2 (0.46) CCR2CCR5CYP2D6CYP2C19
SCHEMBL3855163 0.68 CCR2 (0.46) CCR2CCR5CYP2D6CYP2C19
SCHEMBL14909281 0.68 TSHR (0.30)
SCHEMBL28848429 0.67 CTSS (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1667966-B1 N-ALKYLATED DIAMINOPROPANE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2012-02-29 EP disclosed