SCHEMBL6863742

SCHEMBL6863742

CN(C(=O)c1cc(N)n2nc(-c3ccc(Cl)o3)nc2c1)C1CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 18/20 0.52
MEN1 O00255 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
BLM P54132 1/20 0.42
KMT2A Q03164 1/20 0.42
HSD17B10 Q99714 1/20 0.42
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6871451 0.90 ADORA2A (0.66) ADORA2A
SCHEMBL6863095 0.89 ADORA2A (0.67) ADORA2A
SCHEMBL6869719 0.85 ADORA2A (0.61) ADORA2A
SCHEMBL6863180 0.83 ADORA2A (0.58) ADORA2A
SCHEMBL6867105 0.81 ADORA2A (0.66) ADORA2A
SCHEMBL6863389 0.81 NPC1 (0.47) ADORA2AMEN1MAPTHPGDALOX15
SCHEMBL6871702 0.80 ADORA2A (0.77) ADORA2A
SCHEMBL6869813 0.80 ADORA2A (0.44) ADORA2AMEN1MAPTHPGDALOX15
SCHEMBL6871980 0.80 ADORA2A (0.79) ADORA2A
SCHEMBL6869714 0.79 ADORA2A (0.43) ADORA2AMEN1MAPTHPGDALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US disclosed