SCHEMBL6869714

SCHEMBL6869714

Cc1ccc(-c2nc3cc(C(=O)N(C)C4CCCCC4)cc(N)n3n2)s1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 11/20 0.43
MAPT P10636 2/20 0.43
HPGD P15428 2/20 0.43
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.40
PTAFR P25105 1/20 0.39
KLK7 P49862 1/20 0.38
CNR2 P34972 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
S1PR1 P21453 1/20 0.38
MEN1 O00255 1/20 0.38
ALOX15 P16050 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863785 0.88 ADORA2A (0.44) ADORA2AALDH1A1RAB9A
SCHEMBL6863389 0.83 NPC1 (0.47) ADORA2AMAPTHPGDPOLBPTAFR
SCHEMBL6871451 0.82 ADORA2A (0.66) ADORA2A
SCHEMBL6870443 0.81 LMNA (0.45) ADORA2AMAPTHPGDALDH1A1NPC1
SCHEMBL6869813 0.80 ADORA2A (0.44) ADORA2AMAPTHPGDPOLBNPC1
SCHEMBL6863074 0.80 ADORA2A (0.62) ADORA2AMAPTHPGDALDH1A1POLB
SCHEMBL6870495 0.80 POLB (0.42) ADORA2AMAPTHPGDALDH1A1POLB
SCHEMBL6869707 0.79 KIT (0.44) ADORA2AHPGDALDH1A1POLBNPC1
SCHEMBL6863742 0.79 ADORA2A (0.52) ADORA2AMAPTHPGDPOLBMEN1
SCHEMBL6863095 0.79 ADORA2A (0.67) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed