SCHEMBL6864740

SCHEMBL6864740

O=C(CN1CCN(Cc2ccccc2)CC1)Nc1nc2ccccc2s1

nearest known ligand 0.84

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC27A1 Q6PCB7 1/20 0.67
NFKB1 P19838 1/20 0.64
CSNK1D P48730 1/20 0.64
NFKB2 Q00653 1/20 0.64
RELA Q04206 1/20 0.64
SMN1; SMN2 Q16637 1/20 0.64
PKM P14618 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
CA9 Q16790 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11254394 0.90 PKM (0.59) PKML3MBTL1CA1CA2CA9
SCHEMBL6864105 0.88 SLC27A1 (0.62) SLC27A1NFKB1CSNK1DNFKB2RELA
SCHEMBL6863943 0.88 CLK1 (0.62) SLC27A1SMN1; SMN2
SCHEMBL4806814 0.87 SLC27A1 (0.63) SLC27A1PKML3MBTL1
SCHEMBL8358629 0.87 SLC27A1 (0.63) SLC27A1PKML3MBTL1
SCHEMBL7108865 0.87 SLC27A1 (0.57) SLC27A1
SCHEMBL7522067 0.86 SLC27A1 (0.84) SLC27A1NFKB1CSNK1DNFKB2RELA
SCHEMBL6862327 0.86 SLC27A1 (0.56) SLC27A1NFKB1CSNK1DNFKB2RELA
SCHEMBL6863835 0.86 CSNK1D (0.59) SLC27A1CSNK1DPKML3MBTL1
SCHEMBL6864926 0.85 ALDH1A1 (0.61) SLC27A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US claimed
US-6800444-B1 USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS/INTERMEDIATES ISIS PHARMACEUTICALS, INC. 2004-10-05 US disclosed
US-6660466-B1 Reacting reactive appendage compounds such as meta benzylic compounds or alpha-amide compounds with scaffold molecules having reactive functionalities and contacting the intermediate library with a reducing agent ISIS PHARMACEUTICALS, INC. 2003-12-09 US disclosed
US-6150129-A USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS AND AS INTERMEDIATES FOR PREPARATION OF OTHER PHARMACEUTICAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 2000-11-21 US disclosed
US-5922872-A BACTERICIDES AND DRUGS ISIS PHARMACEUTICALS, INC. (US) 1999-07-13 US disclosed
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US disclosed
US-5798360-A ANTIBACTERIAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 1998-08-25 US disclosed
US-5780241-A ALTERING ELECTROCHEMICAL PROPERTIES BY DECYCLIZATION ISIS PHARMACEUTICALS, INC. (US) 1998-07-14 US disclosed
WO-1998020349-A1 COMPLEX CHEMICAL LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-05-14 WO disclosed
US-5731438-A BACTERICIDES; DRUGS ISIS PHARMACEUTICALS, INC. (US) 1998-03-24 US disclosed