SCHEMBL6866543

SCHEMBL6866543

CCOc1cc(Cc2cnc(N)nc2N)cc(OC(COCc2ccccc2)C2CC2)c1-c1ccc(OC)cc1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.47
CSF1R P07333 1/20 0.47
NTRK3 Q16288 1/20 0.47
NTRK2 Q16620 1/20 0.47
DHFR P00374 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6557380 0.85 NTRK1 (0.64) NTRK1CSF1RNTRK3NTRK2DHFR
SCHEMBL6875102 0.84 DHFR (0.46) DHFR
SCHEMBL6555358 0.84 DHFR (0.48) DHFR
SCHEMBL6556589 0.82 DHFR (0.58) NTRK1CSF1RNTRK3NTRK2DHFR
SCHEMBL6555448 0.82 CSF1R (0.49) NTRK1CSF1RNTRK3NTRK2DHFR
SCHEMBL6556791 0.81 DHFR (0.66) NTRK1CSF1RNTRK3NTRK2DHFR
SCHEMBL7570697 0.80 CSF1R (0.48) NTRK1CSF1RNTRK3NTRK2DHFR
SCHEMBL6874758 0.80 NTRK1 (0.58) NTRK1CSF1RNTRK3NTRK2DHFR
SCHEMBL6555093 0.79 DHFR (0.56) NTRK1CSF1RNTRK3NTRK2DHFR
SCHEMBL6555451 0.79 LMNA (0.58) NTRK1CSF1RNTRK3NTRK2DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6821980-B1 Substituted 5-benzyl-2,4-diaminopyrimidines BASILEA PHARMACEUTICA AG (CH) 2004-11-23 US disclosed
EP-1230224-A1 SUBSTITUTED 5-BENZYL-2,4-DIAMINOPYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 2002-08-14 EP disclosed
WO-2001032633-A1 SUBSTITUTED 5-BENZYL-2,4-DIAMINOPYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2001-05-10 WO disclosed