SCHEMBL6867360

SCHEMBL6867360

COCCN(C[C@H]1CC[C@@H](Nc2nccc(N(C)C)n2)CC1)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.39
MCHR1 Q99705 14/20 0.39
CNR1 P21554 1/20 0.38
KCNH2 Q12809 1/20 0.38
AURKB Q96GD4 1/20 0.38
DRD2 P14416 1/20 0.37
ADRA2A P08913 4/20 0.37
HRH1 P35367 4/20 0.37
HTR2B P41595 4/20 0.37
ADRA1A P35348 2/20 0.37
BCHE P06276 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867366 1.00 MAPK14 (0.39) MAPK14MCHR1CNR1KCNH2AURKB
SCHEMBL6879155 0.87 DRD2 (0.42) MAPK14DRD2
SCHEMBL6879152 0.87 DRD2 (0.42) MAPK14DRD2
SCHEMBL6868816 0.84 CNR1 (0.39) MAPK14MCHR1CNR1KCNH2AURKB
SCHEMBL6873416 0.84 MAPK14 (0.40) MAPK14MCHR1DRD2ADRA2AHRH1
SCHEMBL6873422 0.84 MAPK14 (0.40) MAPK14MCHR1DRD2ADRA2AHRH1
SCHEMBL6879294 0.83 MAPK14 (0.40) MAPK14MCHR1DRD2ADRA2AHRH1
SCHEMBL6879291 0.83 MAPK14 (0.40) MAPK14MCHR1DRD2ADRA2AHRH1
SCHEMBL6867607 0.80 MAPK8 (0.39) MAPK14MCHR1DRD2
SCHEMBL6867614 0.80 MAPK8 (0.39) MAPK14MCHR1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed