SCHEMBL6868816

SCHEMBL6868816

COCCN(C(=O)O)[C@H]1CC[C@@H](Nc2nccc(N(C)C)n2)CC1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.39
KCNH2 Q12809 1/20 0.39
AURKB Q96GD4 1/20 0.39
MCHR1 Q99705 14/20 0.39
ADRA2A P08913 4/20 0.38
HRH1 P35367 4/20 0.38
HTR2B P41595 3/20 0.38
ADRA1A P35348 2/20 0.38
LCK P06239 1/20 0.37
JAK3 P52333 1/20 0.37
MAPK14 Q16539 2/20 0.37
MAPK8 P45983 1/20 0.35
MAPK9 P45984 1/20 0.35
MAPK10 P53779 1/20 0.35
SMYD3 Q9H7B4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6877440 0.87 MAPK8 (0.40) MCHR1JAK3MAPK14MAPK8MAPK9
SCHEMBL6877450 0.87 MAPK8 (0.40) MCHR1JAK3MAPK14MAPK8MAPK9
SCHEMBL6867366 0.84 MAPK14 (0.39) CNR1KCNH2AURKBMCHR1ADRA2A
SCHEMBL6867360 0.84 MAPK14 (0.39) CNR1KCNH2AURKBMCHR1ADRA2A
SCHEMBL6878045 0.83 HRH4 (0.42) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6878052 0.83 HRH4 (0.42) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6877753 0.82 LCK (0.39) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6877758 0.82 LCK (0.39) MCHR1ADRA2AHRH1HTR2BADRA1A
SCHEMBL6877016 0.79 MAPK8 (0.39) AURKBMCHR1ADRA2AHRH1HTR2B
SCHEMBL6877019 0.79 MAPK8 (0.39) AURKBMCHR1ADRA2AHRH1HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed