SCHEMBL6867674

SCHEMBL6867674

Cc1cc([N+](=O)[O-])ccc1NC(=O)N[C@H]1CC[C@@H](Nc2nc3c(c(N(C)C)n2)CCCC3)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.47
MCHR1 Q99705 2/20 0.47
LMNA P02545 5/20 0.46
MAPT P10636 5/20 0.46
ALDH1A1 P00352 4/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
RAB9A P51151 3/20 0.43
NPC1 O15118 2/20 0.43
POLB P06746 1/20 0.43
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
HTT P42858 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MAPK1 P28482 1/20 0.40
TRPV1 Q8NER1 1/20 0.39
EPHX1 P07099 1/20 0.39
HRH1 P35367 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867680 1.00 ADRA2A (0.47) ADRA2AMCHR1LMNAMAPTALDH1A1
SCHEMBL6873005 0.93 MCHR1 (0.47) ADRA2AMCHR1LMNAMAPTALDH1A1
SCHEMBL6873000 0.93 MCHR1 (0.47) ADRA2AMCHR1LMNAMAPTALDH1A1
SCHEMBL6873523 0.92 ADRA2A (0.46) ADRA2AMCHR1LMNAMAPTALDH1A1
SCHEMBL6873527 0.92 ADRA2A (0.46) ADRA2AMCHR1LMNAMAPTALDH1A1
SCHEMBL6879371 0.91 KMT2A (0.53) ADRA2AMCHR1LMNAMAPTALDH1A1
SCHEMBL6879376 0.91 KMT2A (0.53) ADRA2AMCHR1LMNAMAPTALDH1A1
SCHEMBL6873049 0.91 ALDH1A1 (0.45) ADRA2AMCHR1LMNAMAPTALDH1A1
SCHEMBL6873057 0.91 ALDH1A1 (0.45) ADRA2AMCHR1LMNAMAPTALDH1A1
SCHEMBL6878618 0.89 NPSR1 (0.48) ADRA2AMCHR1LMNAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed