SCHEMBL6868029

SCHEMBL6868029

Cc1ccsc1-c1nc2cc(C(=O)NC3CCc4ccccc43)cc(N)n2n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 4/20 0.52
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
TAS1R3 Q7RTX0 2/20 0.42
TAS1R1 Q7RTX1 2/20 0.42
CNR1 P21554 3/20 0.42
CNR2 P34972 1/20 0.42
HPGDS O60760 1/20 0.42
LMNA P02545 2/20 0.41
KDM4E B2RXH2 2/20 0.41
USP2 O75604 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
HTT P42858 1/20 0.41
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6873668 0.85 CHRM4 (0.47) CHRM4PDE4APDE4BPDE4CPDE4D
SCHEMBL6863240 0.84 CHRM4 (0.55) CHRM4PDE4APDE4BPDE4CPDE4D
SCHEMBL6870587 0.84 CHRM4 (0.49) CHRM4PDE4APDE4BPDE4CPDE4D
SCHEMBL6872383 0.82 ADORA2A (0.56) CHRM4PDE4APDE4BPDE4CPDE4D
SCHEMBL6870459 0.81 ADORA2A (0.43) TAS1R3TAS1R1LMNAKDM4ECYP1A2
SCHEMBL6863147 0.79 CHRM4 (0.46) CHRM4PDE4APDE4BPDE4CPDE4D
SCHEMBL6870464 0.78 ADORA2A (0.42) LMNACYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL6867741 0.75 ADORA2A (0.46) KDM4EHTTALDH1A1HPGD
SCHEMBL6871970 0.75 ADORA2A (0.43) HPGD
SCHEMBL6872082 0.73 KMT2A (0.51) CHRM4LMNAKDM4ECYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed