SCHEMBL6870587

SCHEMBL6870587

Nc1cc(C(=O)NC2CCc3ccccc32)cc2nc(-c3ccccc3)nn12

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 3/20 0.49
HTT P42858 1/20 0.47
HPGDS O60760 1/20 0.46
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
CFD P00746 2/20 0.44
CNR1 P21554 2/20 0.44
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44
BRD4 O60885 1/20 0.43
ROCK2 O75116 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
KMT2A Q03164 1/20 0.43
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6863147 0.89 CHRM4 (0.46) CHRM4HTTHPGDSPDE4APDE4B
SCHEMBL6863240 0.85 CHRM4 (0.55) CHRM4HTTHPGDSPDE4APDE4B
SCHEMBL6873668 0.85 CHRM4 (0.47) CHRM4HTTHPGDSPDE4APDE4B
SCHEMBL6872383 0.85 ADORA2A (0.56) CHRM4HPGDSPDE4APDE4BPDE4C
SCHEMBL6868029 0.84 CHRM4 (0.52) CHRM4HTTHPGDSPDE4APDE4B
SCHEMBL7708892 0.82 FADS1 (0.43) CHRM4HTTKDM4EMEN1ALDH1A1
SCHEMBL6868095 0.81 KDM4E (0.53) HTTCNR1KDM4EMEN1ALDH1A1
SCHEMBL7711667 0.76 MAPK13 (0.43) HTTCNR1MEN1KMT2A
SCHEMBL6868100 0.75 ADORA2A (0.44) HTTKDM4EMEN1ALDH1A1HPGD
SCHEMBL6870681 0.74 ADORA2A (0.49) HTTKDM4EMEN1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed