SCHEMBL6863240

SCHEMBL6863240

Cc1ccc(-c2nc3cc(C(=O)NC4CCc5ccccc54)cc(N)n3n2)s1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 5/20 0.55
TAS1R3 Q7RTX0 3/20 0.47
TAS1R1 Q7RTX1 3/20 0.47
CNR1 P21554 3/20 0.45
CNR2 P34972 1/20 0.45
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HPGDS O60760 1/20 0.43
LMNA P02545 2/20 0.43
HTT P42858 2/20 0.42
USP2 O75604 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870587 0.85 CHRM4 (0.49) CHRM4TAS1R3TAS1R1CNR1PDE4A
SCHEMBL6868029 0.84 CHRM4 (0.52) CHRM4TAS1R3TAS1R1CNR1CNR2
SCHEMBL6872383 0.83 ADORA2A (0.56) CHRM4PDE4APDE4BPDE4CPDE4D
SCHEMBL6873668 0.82 CHRM4 (0.47) CHRM4TAS1R3TAS1R1CNR1PDE4A
SCHEMBL6863147 0.81 CHRM4 (0.46) CHRM4TAS1R3TAS1R1CNR1PDE4A
SCHEMBL6870443 0.81 LMNA (0.45) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL6870449 0.77 RAB9A (0.45) ALDH1A1HPGDMEN1KMT2ALMNA
SCHEMBL6863351 0.75 PLAU (0.47) CHRM4KDM4EALDH1A1HPGDMEN1
SCHEMBL6871437 0.74 ADORA2A (0.47) ALDH1A1HPGDHTT
SCHEMBL6868343 0.74 ADORA2A (0.45) KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed